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Wiley电子期刊(1)
NATURE电子期刊(6)
ACS电子期刊(13)
SpringerLink电子期刊(4)
Elsevier电子期刊(38)
在“
ACS电子期刊
”中,
命中:
13
条,耗时:小于0.01 秒
在所有数据库中总计命中:
62
条
1.
Docking and Linking of Fragments To Discover Jumonji Histone Demethylase Inhibitors
作者:
Magdalena Korczynska
;
Daniel D. Le
;
Noah Younger
;
Elisabet Gregori-Puigjané
;
Anthony Tumber
;
Tobias Krojer
;
Srikannathasan Velupillai
;
Carina Gileadi
;
Radosław P. Nowak
;
Eriko Iwasa
;
Samuel B. Pollock
;
Idelisse Ortiz Torres
;
Udo
Oppermann
;
Brian K. Shoichet
;
Danica Galonić Fujimori
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors
作者:
Vassilios Bavetsias
;
Rachel M. Lanigan
;
Gian Filippo Ruda
;
Butrus Atrash
;
Mark G. McLaughlin
;
Anthony Tumber
;
N. Yi Mok
;
Yann-Vaï Le Bihan
;
Sally Dempster
;
Katherine J. Boxall
;
Fiona Jeganathan
;
Stephanie B. Hatch
;
Pavel Savitsky
;
Srikannathasan Velupillai
;
Tobias Krojer
;
Katherine S. England
;
Jimmy Sejberg
;
Ching Thai
;
Adam Donovan
;
Akos Pal
;
Giuseppe Scozzafava
;
James M. Bennett
;
Akane Kawamura
;
Catrine Johansson
;
Aleksandra Szykowska
;
Carina Gileadi
;
Nicola A. Burgess-Brown
;
Frank von Delft
;
Udo
Oppermann
;
Zoe Walters
;
Janet Shipley
;
Florence I. Raynaud
;
Susan M. Westaway
;
Rab K. Prinjha
;
Oleg Fedorov
;
Rosemary Burke
;
Christopher J. Schofield
;
Isaac M. Westwood
;
Chas Bountra
;
Susanne Müller
;
Rob L. M. van Montfort
;
Paul E. Brennan
;
Julian Blagg
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Discovery of NCT-501, a Potent and Selective Theophylline-Based Inhibitor of Aldehyde Dehydrogenase 1A1 (ALDH1A1)
作者:
Shyh-Ming Yang
;
Adam Yasgar
;
Bettina Miller
;
Madhu Lal-Nag
;
Kyle Brimacombe
;
Xin Hu
;
Hongmao Sun
;
Amy Wang
;
Xin Xu
;
Kimloan Nguyen
;
Udo
Oppermann
;
Marc Ferrer
;
Vasilis Vasiliou
;
Anton Simeonov
;
Ajit Jadhav
;
David J. Maloney
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Quantitative Analysis of Histone Demethylase Probes Using Fluorescence Polarization
作者:
Wenqing Xu
;
Jessica D. Podoll
;
Xuan Dong
;
Anthony Tumber
;
Udo
Oppermann
;
Xiang Wang
刊名:Journal of Medicinal Chemistry
出版年:2013
5.
Structure of MMACHC Reveals an Arginine-Rich Pocket and a Domain-Swapped Dimer for Its B12 Processing Function
作者:
D. Sean Froese
;
Tobias Krojer
;
Xuchu Wu
;
Roshi Shrestha
;
Wasim Kiyani
;
Frank von Delft
;
Roy A. Gravel
;
Udo
Oppermann
;
Wyatt W. Yue
刊名:Biochemistry
出版年:2012
6.
Plant Growth Regulator Daminozide Is a Selective Inhibitor of Human KDM2/7 Histone Demethylases
作者:
Nathan R. Rose
;
Esther C. Y. Woon
;
Anthony Tumber
;
Louise J. Walport
;
Rasheduzzaman Chowdhury
;
Xuan Shirley Li
;
Oliver N. F. King
;
Clarisse Lejeune
;
Stanley S. Ng
;
Tobias Krojer
;
Mun Chiang Chan
;
Anna M. Rydzik
;
Richard J. Hopkinson
;
Ka Hing Che
;
Michelle Daniel
;
Claire Strain-Damerell
;
Carina Gileadi
;
Grazyna Kochan
;
Ivanhoe K. H. Leung
;
James Dunford
;
Kar Kheng Yeoh
;
Peter J. Ratcliffe
;
Nicola Burgess-Brown
;
Frank von Delft
;
Susanne Muller
;
Brian Marsden
;
Paul E. Brennan
;
Michael A. McDonough
;
Udo
Oppermann
;
Robert J. Klose
;
Christopher J. Schofield
;
Akane Kawamura
刊名:Journal of Medicinal Chemistry
出版年:2012
7.
A Selective Inhibitor and Probe of the Cellular Functions of Jumonji C Domain-Containing Histone Demethylases
作者:
Xuelai Luo
;
Yongxiang Liu
;
Stefan Kubicek
;
Johanna Myllyharju
;
Anthony Tumber
;
Stanley Ng
;
Ka Hing Che
;
Jessica Podoll
;
Tom D. Heightman
;
Udo
Oppermann
;
Stuart L. Schreiber
;
Xiang Wang
刊名:Journal of the American Chemical Society
出版年:2011
8.
Selective Inhibitors of the JMJD2 Histone Demethylases: Combined Nondenaturing Mass Spectrometric Screening and Crystallographic Approaches
作者:
Nathan R. Rose
;
Esther C. Y. Woon
;
Guy L. Kingham
;
Oliver N. F. King
;
Jasmin Mecinovi
;
Ian J. Clifton
;
Stanley S. Ng
;
Jobina Talib-Hardy
;
Udo
Oppermann
;
Michael A. McDonough
;
Christopher J. Schofield
刊名:Journal of Medicinal Chemistry
出版年:2010
9.
Structural Impact of Human and Escherichia coli Biotin Carboxyl Carrier Proteins on Biotin Attachment
作者:
Shannon Healy
;
Megan K. McDonald
;
Xuchu Wu
;
Wyatt W. Yue
;
Grazyna Kochan
;
Udo
Oppermann
;
Roy A. Gravel
刊名:Biochemistry
出版年:2010
10.
SALMON: Solvent Accessibility, Ligand binding, and Mapping of ligand Orientation by NMR Spectroscopy
作者:
Christian Ludwig
;
Paul J. A. Michiels
;
Xiaoqiu Wu
;
Kathryn L. Kavanagh
;
Ewa Pilka
;
Anna Jansson
;
Udo
Oppermann
;
Ulrich L. Gü
;
nther
刊名:Journal of Medicinal Chemistry
出版年:2008
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