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ACS电子期刊(15)
在“
ACS电子期刊
”中,
命中:
15
条,耗时:小于0.01 秒
在所有数据库中总计命中:
53
条
1.
Fragment Molecular Orbital Method Applied to Lead Optimization of Novel Interleukin-2 Inducible T-Cell Kinase (ITK) Inhibitors
作者:
Alexander Heifetz
;
Giancarlo Trani
;
Matteo Aldeghi
;
Colin H. MacKinnon
;
Paul A. McEwan
;
Frederick A. Brookfield
;
Ewa I. Chudyk
;
Mike Bodkin
;
Zhonghua
Pei
;
Jason D. Burch
;
Daniel F. Ortwine
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Linker Immolation Determines Cell Killing Activity of Disulfide-Linked Pyrrolobenzodiazepine Antibody–Drug Conjugates
作者:
Donglu Zhang
;
Thomas H. Pillow
;
Yong Ma
;
Josefa dela Cruz-Chuh
;
Katherine R. Kozak
;
Jack D. Sadowsky
;
Gail D. Lewis Phillips
;
Jun Guo
;
Martine Darwish
;
Peter Fan
;
Jingtian Chen
;
Changrong He
;
Tao Wang
;
Hui Yao
;
Zijin Xu
;
Jinhua Chen
;
John Wai
;
Zhonghua
Pei
;
Cornelis E. C. A. Hop
;
S. Cyrus Khojasteh
;
Peter S. Dragovich
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Comparative Study of Nonautolytic Mutant and Wild-Type Strains of Coprinopsis cinerea Supports an Important Role of Glucanases in Fruiting Body Autolysis
作者:
Zhonghua
Liu
;
Xin Niu
;
Jun Wang
;
Wenming Zhang
;
Mingmei Yang
;
Cuicui Liu
;
Yuanjing Xiong
;
Yan Zhao
;
Siyu
Pei
;
Qin Qin
;
Yu Zhang
;
Yuan Yu
;
Sheng Yuan
刊名:Journal of Agricultural and Food Chemistry
出版年:2015
4.
Tetrahydroindazoles as Interleukin-2 Inducible T-Cell Kinase Inhibitors. Part II. Second-Generation Analogues with Enhanced Potency, Selectivity, and Pharmacodynamic Modulation in Vivo
作者:
Jason D. Burch
;
Kathy Barrett
;
Yuan Chen
;
Jason DeVoss
;
Charles Eigenbrot
;
Richard Goldsmith
;
M. Hicham A. Ismaili
;
Kevin Lau
;
Zhonghua
Lin
;
Daniel F. Ortwine
;
Ali A. Zarrin
;
Paul A. McEwan
;
John J. Barker
;
Claire Ellebrandt
;
Daniel Kordt
;
Daniel B. Stein
;
Xiaolu Wang
;
Yong Chen
;
Baihua Hu
;
Xiaofeng Xu
;
Po-Wai Yuen
;
Yamin Zhang
;
Zhonghua
Pei
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Property- and Structure-Guided Discovery of a Tetrahydroindazole Series of Interleukin-2 Inducible T-Cell Kinase Inhibitors
作者:
Jason D. Burch
;
Kevin Lau
;
John J. Barker
;
Fred Brookfield
;
Yong Chen
;
Yuan Chen
;
Charles Eigenbrot
;
Claire Ellebrandt
;
M. Hicham A. Ismaili
;
Adam Johnson
;
Daniel Kordt
;
Colin H. MacKinnon
;
Paul A. McEwan
;
Daniel F. Ortwine
;
Daniel B. Stein
;
Xiaolu Wang
;
Dirk Winkler
;
Po-Wai Yuen
;
Yamin Zhang
;
Ali A. Zarrin
;
Zhonghua
Pei
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
Discovery and Biological Profiling of Potent and Selective mTOR Inhibitor GDC-0349
作者:
Zhonghua
Pei
;
Elizabeth Blackwood
;
Lichuan Liu
;
Shiva Malek
;
Marcia Belvin
;
Michael F. T. Koehler
;
Daniel F. Ortwine
;
Huifen Chen
;
Frederick Cohen
;
Jane R. Kenny
;
Philippe Bergeron
;
Kevin Lau
;
Cuong Ly
;
Xianrui Zhao
;
Anthony A. Estrada
;
Tom Truong
;
Jennifer A. Epler
;
Jim Nonomiya
;
Lan Trinh
;
Steve Sideris
;
John Lesnick
;
Linda Bao
;
Ulka Vijapurkar
;
Sophie Mukadam
;
Suzanne Tay
;
Gauri Deshmukh
;
Yung-Hsiang Chen
;
Xiao Ding
;
Lori S. Friedman
;
Joseph P. Lyssikatos
刊名:ACS Medicinal Chemistry Letters
出版年:2013
7.
Pyrimidoaminotropanes as Potent, Selective, and Efficacious Small Molecule Kinase Inhibitors of the Mammalian Target of Rapamycin (mTOR)
作者:
Anthony A. Estrada
;
Daniel G. Shore
;
Elizabeth Blackwood
;
Yung-Hsiang Chen
;
Gauri Deshmukh
;
Xiao Ding
;
Antonio G. DiPasquale
;
Jennifer A. Epler
;
Lori S. Friedman
;
Michael F. T. Koehler
;
Lichuan Liu
;
Shiva Malek
;
Jim Nonomiya
;
Daniel F. Ortwine
;
Zhonghua
Pei
;
Steve Sideris
;
Frederic St-Jean
;
Lan Trinh
;
Tom Truong
;
Joseph P. Lyssikatos
刊名:Journal of Medicinal Chemistry
出版年:2013
8.
Potent, Selective, and Orally Bioavailable Inhibitors of the Mammalian Target of Rapamycin Kinase Domain Exhibiting Single Agent Antiproliferative Activity
作者:
Michael F. T. Koehler
;
Philippe Bergeron
;
Elizabeth Blackwood
;
Krista K. Bowman
;
Yung-Hsiang Chen
;
Gauri Deshmukh
;
Xiao Ding
;
Jennifer Epler
;
Kevin Lau
;
Leslie Lee
;
Lichuan Liu
;
Cuong Ly
;
Shiva Malek
;
Jim Nonomiya
;
Jason Oeh
;
Daniel F. Ortwine
;
Deepak Sampath
;
Steve Sideris
;
Lan Trinh
;
Tom Truong
;
Jiansheng Wu
;
Zhonghua
Pei
;
Joseph P. Lyssikatos
刊名:Journal of Medicinal Chemistry
出版年:2012
9.
Femtosecond Time-Resolved Fluorescence Study of TiO2-Coated ZnO Nanorods/P3HT Photovoltaic Films
作者:
Yong Li
;
Pei
fen Lu
;
Minlin Jiang
;
Rabin Dhakal
;
Prem Thapaliya
;
Zhonghua
Peng
;
Binay Jha
;
Xingzhong Yan
刊名:The Journal of Physical Chemistry C
出版年:2012
10.
Potent, Selective, and Orally Bioavailable Inhibitors of Mammalian Target of Rapamycin (mTOR) Kinase Based on a Quaternary Substituted Dihydrofuropyrimidine
作者:
Frederick Cohen
;
Philippe Bergeron
;
Elizabeth Blackwood
;
Krista K. Bowman
;
Huifen Chen
;
Antonio G. DiPasquale
;
Jennifer A. Epler
;
Michael F. T. Koehler
;
Kevin Lau
;
Cristina Lewis
;
Lichuan Liu
;
Cuong Q. Ly
;
Shiva Malek
;
Jim Nonomiya
;
Daniel F. Ortwine
;
Zhonghua
Pei
;
Kirk D. Robarge
;
Steve Sideris
;
Lan Trinh
;
Tom Truong
;
Jiansheng Wu
;
Xianrui Zhao
;
Joseph P. Lyssikatos
刊名:Journal of Medicinal Chemistry
出版年:2011
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