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Elsevier电子期刊(21)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
31
条
1.
Determination of Antibody–Drug Conjugate Released Payload Species Using Directed in Vitro Assays and Mass Spectrometric Interrogation
作者:
Andrew J. Bessire
;
T. Eric Ballard
;
Manoj Charati
;
Justin Cohen
;
Michael Green
;
My-Hanh Lam
;
Frank Loganzo
;
Birte Nolting
;
Betsy Pierce
;
Sujiet Puthenveetil
;
Lee Roberts
;
Klaas Schildknegt
;
Chakrapani
Subramanyam
刊名:Bioconjugate Chemistry
出版年:2016
2.
Natural Product Splicing Inhibitors: A New Class of Antibody–Drug Conjugate (ADC) Payloads
作者:
Sujiet Puthenveetil
;
Frank Loganzo
;
Haiyin He
;
Ken Dirico
;
Michael Green
;
Jesse Teske
;
Sylvia Musto
;
Tracey Clark
;
Brian Rago
;
Frank Koehn
;
Robert Veneziale
;
Hadi Falahaptisheh
;
Xiaogang Han
;
Frank Barletta
;
Judy Lucas
;
Chakrapani
Subramanyam
;
Christopher J. O’Donnell
;
L. Nathan Tumey
;
Puja Sapra
;
Hans Peter Gerber
;
Dangshe Ma
;
Edmund I. Graziani
刊名:Bioconjugate Chemistry
出版年:2016
3.
Design, Synthesis, and Cytotoxic Evaluation of Novel Tubulysin Analogues as ADC Payloads
作者:
Carolyn A. Leverett
;
Sai Chetan K. Sukuru
;
Beth C. Vetelino
;
Sylvia Musto
;
Kevin Parris
;
Jayvardhan Pandit
;
Frank Loganzo
;
Alison H. Varghese
;
Guoyun Bai
;
Bin Liu
;
Dingguo Liu
;
Sarah Hudson
;
Venkata Ramana Doppalapudi
;
Joseph Stock
;
Christopher J. O’Donnell
;
Chakrapani
Subramanyam
刊名:ACS Medicinal Chemistry Letters
出版年:2016
4.
Optimization of Tubulysin Antibody–Drug Conjugates: A Case Study in Addressing ADC Metabolism
作者:
L. Nathan Tumey
;
Carolyn A. Leverett
;
Beth Vetelino
;
Fengping Li
;
Brian Rago
;
Xiaogang Han
;
Frank Loganzo
;
Sylvia Musto
;
Guoyun Bai
;
Sai Chetan K. Sukuru
;
Edmund I. Graziani
;
Sujiet Puthenveetil
;
Jeffrey Casavant
;
Anokha Ratnayake
;
Kimberly Marquette
;
Sarah Hudson
;
Venkata Ramana Doppalapudi
;
Joseph Stock
;
Lioudmila Tchistiakova
;
Andrew J. Bessire
;
Tracey Clark
;
Judy Lucas
;
Christine Hosselet
;
Christopher J. O’Donnell
;
Chakrapani
Subramanyam
刊名:ACS Medicinal Chemistry Letters
出版年:2016
5.
Design of Pyridopyrazine-1,6-dione 纬-Secretase Modulators that Align Potency, MDR Efflux Ratio, and Metabolic Stability
作者:
Martin Pettersson
;
Douglas S. Johnson
;
John M. Humphrey
;
Todd W. Butler
;
Christopher W. am Ende
;
Benjamin A. Fish
;
Michael E. Green
;
Gregory W. Kauffman
;
Patrick B. Mullins
;
Christopher J. O鈥橠onnell
;
Antonia F. Stepan
;
Cory M. Stiff
;
Chakrapani
Subramanyam
;
Tuan P. Tran
;
Beth Cooper Vetelino
;
Eddie Yang
;
Longfei Xie
;
Kelly R. Bales
;
Leslie R. Pustilnik
;
Stefanus J. Steyn
;
Kathleen M. Wood
;
Patrick R. Verhoest
刊名:ACS Medicinal Chemistry Letters
出版年:2015
6.
Design, Synthesis, and Pharmacological Evaluation of a Novel Series of Pyridopyrazine-1,6-dione γ-Secretase Modulators
作者:
Martin Pettersson
;
Douglas S. Johnson
;
Chakrapani
Subramanyam
;
Kelly R. Bales
;
Christopher W. am Ende
;
Benjamin A. Fish
;
Michael E. Green
;
Gregory W. Kauffman
;
Patrick B. Mullins
;
Thayalan Navaratnam
;
Subas M. Sakya
;
Cory M. Stiff
;
Tuan P. Tran
;
Longfei Xie
;
Liming Zhang
;
Leslie R. Pustilnik
;
Beth C. Vetelino
;
Kathleen M. Wood
;
Nikolay Pozdnyakov
;
Patrick R. Verhoest
;
Christopher J. O’Donnell
刊名:Journal of Medicinal Chemistry
出版年:2014
7.
Discovery of Cytotoxic Dolastatin 10 Analogues with N-Terminal Modifications
作者:
Andreas Maderna
;
Matthew Doroski
;
Chakrapani
Subramanyam
;
Alexander Porte
;
Carolyn A. Leverett
;
Beth C. Vetelino
;
Zecheng Chen
;
Hud Risley
;
Kevin Parris
;
Jayvardhan Pandit
;
Alison H. Varghese
;
Suman Shanker
;
Cynthia Song
;
Sai Chetan K. Sukuru
;
Kathleen A. Farley
;
Melissa M. Wagenaar
;
Michael J. Shapiro
;
Sylvia Musto
;
My-Hanh Lam
;
Frank Loganzo
;
Christopher J. O鈥橠onnell
刊名:Journal of Medicinal Chemistry
出版年:2014
8.
Ligand鈥揚rotein Interactions of Selective Casein Kinase 1未 Inhibitors
作者:
Scot Mente
;
Eric Arnold
;
Todd Butler
;
Subramanyam
Chakrapani
;
Ramalakshmi Chandrasekaran
;
Kevin Cherry
;
Ken DiRico
;
Angela Doran
;
Katherine Fisher
;
Paul Galatsis
;
Michael Green
;
Matthew Hayward
;
John Humphrey
;
John Knafels
;
Jianke Li
;
Shenping Liu
;
Michael Marconi
;
Scott McDonald
;
Jeff Ohren
;
Vanessa Paradis
;
Blossom Sneed
;
Kevin Walton
;
Travis Wager
刊名:Journal of Medicinal Chemistry
出版年:2013
9.
Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active 纬-Secretase Inhibitor
作者:
Antonia F. Stepan
;
Chakrapani
Subramanyam
;
Ivan V. Efremov
;
Jason K. Dutra
;
Theresa J. O鈥橲ullivan
;
Kenneth J. DiRico
;
W. Scott McDonald
;
Annie Won
;
Peter H. Dorff
;
Charles E. Nolan
;
Stacey L. Becker
;
Leslie R. Pustilnik
;
David R. Riddell
;
Gregory W. Kauffman
;
Bethany L. Kormos
;
Liming Zhang
;
Yasong Lu
;
Steven H. Capetta
;
Michael E. Green
;
Kapil Karki
;
Evelyn Sibley
;
Kevin P. Atchison
;
Andrew J. Hallgren
;
Christine E. Oborski
;
Ashley E. Robshaw
;
Blossom Sneed
;
Christopher J. O鈥橠onnell
刊名:Journal of Medicinal Chemistry
出版年:2012
10.
Metabolism-Directed Design of Oxetane-Containing Arylsulfonamide Derivatives as 纬-Secretase Inhibitors
作者:
Antonia F. Stepan
;
Kapil Karki
;
W. Scott McDonald
;
Peter H. Dorff
;
Jason K. Dutra
;
Kenneth J. DiRico
;
Annie Won
;
Chakrapani
Subramanyam
;
Ivan V. Efremov
;
Christopher J. O鈥橠onnell
;
Charles E. Nolan
;
Stacey L. Becker
;
Leslie R. Pustilnik
;
Blossom Sneed
;
Hao Sun
;
Yasong Lu
;
Ashley E. Robshaw
;
David Riddell
;
Theresa J. O'Sullivan
;
Evelyn Sibley
;
Steven Capetta
;
Kevin Atchison
;
Andrew J. Hallgren
;
Emily Miller
;
Anthony Wood
;
R. Scott Obach
刊名:Journal of Medicinal Chemistry
出版年:2011
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