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SpringerLink电子期刊(1)
NATURE电子期刊(1)
Elsevier电子期刊(10)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
22
条
1.
Disc
o
very
o
f a P
o
tent Acyclic, Tripeptidic, Acyl Sulf
o
namide Inhibit
o
r
o
f Hepatitis C Virus NS3 Pr
o
tease as a Back-up t
o
Asunaprevir with the P
o
tential f
o
r Once-Daily D
o
sing
作者:
Li-Qiang Sun
;
Eric Mull
;
Barbara Zheng
;
Stanley D’Andrea
;
Qian Zha
o
;
Alan Xiangd
o
ng Wang
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Jie Chen
;
Anth
o
ny C
o
cuzza
;
D
o
nna M. Bilder
;
Arvind Mathur
;
Richard Rampulla
;
Bang-Chi Chen
;
Theerthagiri Palani
;
Sivakumar Ganesan
;
Pirama Nayagam Arunachalam
;
Paul Falk
;
Steven Levine
;
Cha
o
qun Chen
;
Jacques Frib
o
rg
;
Fei Yu
;
Dennis Hernandez
;
Amy K. Sheaffer
;
Jay
O
.
Knipe
;
Y
o
ng-Hae Han
;
Richard Schartman
;
Maria D
o
n
o
s
o
;
Kathy M
o
sure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Ramkumar Rajamani
;
Kevin Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Ga
o
;
Alicia Ng
;
Lucian
o
Mueller
;
Dennis M. Grasela
;
Stephen Adams
;
James L
o
y
;
Paul C. Levesque
;
Huabin Sun
;
H
o
ng Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jial
o
ng Zhu
;
Ying-Kai Wang
;
Hua Fang
;
Mark I. C
o
ckett
;
Nich
o
las A. Meanwell
;
Fi
o
na McPhee
;
Paul M. Sc
o
la
刊名:J
o
urnal
o
f Medicinal Chemistry
出版年:2016
2.
Hepatitis C Virus NS5A Replicati
o
n C
o
mplex Inhibit
o
rs. Part 6: Disc
o
very
o
f a N
o
vel and Highly P
o
tent Biarylimidaz
o
le Chem
o
type with Inhibit
o
ry Activity T
o
ward Gen
o
types 1a and 1b Replic
o
ns
作者:
Mak
o
nen Belema
;
Van N. Nguyen
;
Jeffrey L. R
o
mine
;
Denis R. St. Laurent
;
O
mar D. L
o
pez
;
Jas
o
n T. G
oo
drich
;
Peter T. N
o
wer
;
D
o
nald R. O鈥橞
o
yle
;
II
;
Julie A. Lemm
;
R
o
bert A. Fridell
;
Min Ga
o
;
Hua Fang
;
Rud
o
lph G. Krause
;
Ying-Kai Wang
;
A.
Jay
ne
O
liver
;
Andrew C. G
oo
d
;
Jay
O
.
Knipe
;
Nich
o
las A. Meanwell
;
Lawrence B. Snyder
刊名:J
o
urnal
o
f Medicinal Chemistry
出版年:2014
3.
Hepatitis C Virus NS5A Replicati
o
n C
o
mplex Inhibit
o
rs: The Disc
o
very
o
f Daclatasvir
作者:
Mak
o
nen Belema
;
Van N. Nguyen
;
Car
o
l Bachand
;
Dan H. De
o
n
;
Jas
o
n T. G
oo
drich
;
Clint A. James
;
Ric
o
Lav
o
ie
;
O
mar D. L
o
pez
;
Alain Martel
;
Jeffrey L. R
o
mine
;
Edward H. Ruediger
;
Lawrence B. Snyder
;
Denis R. St. Laurent
;
Fukang Yang
;
Juliang Zhu
;
Henry S. W
o
ng
;
David R. Langley
;
Stephen P. Adams
;
Glenn H. Cant
o
r
;
Anjaneya Chimalak
o
nda
;
Aberra Fura
;
Benjamin M. J
o
hns
o
n
;
Jay
O
.
Knipe
;
Dawn D. Parker
;
Kenneth S. Sant
o
ne
;
R
o
bert A. Fridell
;
Julie A. Lemm
;
D
o
nald R. O鈥橞
o
yle
;
II
;
Richard J. C
o
l
o
nn
o
;
Min Ga
o
;
Nich
o
las A. Meanwell
;
Lawrence G. Hamann
刊名:J
o
urnal
o
f Medicinal Chemistry
出版年:2014
4.
Disc
o
very and Early Clinical Evaluati
o
n
o
f BMS-605339, a P
o
tent and Orally Efficaci
o
us Tripeptidic Acylsulf
o
namide NS3 Pr
o
tease Inhibit
o
r f
o
r the Treatment
o
f Hepatitis C Virus Infecti
o
n
作者:
Paul M. Sc
o
la
;
Alan Xiangd
o
ng Wang
;
Andrew C. G
oo
d
;
Li-Qiang Sun
;
Keith D. C
o
mbrink
;
Jeffrey A. Campbell
;
Jie Chen
;
Y
o
ng Tu
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Anth
o
ny C
o
cuzza
;
D
o
nna M. Bilder
;
Stanley D鈥橝ndrea
;
Barbara Zheng
;
Piyasena Hewawasam
;
Min Ding
;
Jan Thuring
;
Jianqing Li
;
Dennis Hernandez
;
Fei Yu
;
Paul Falk
;
Guangzhi Zhai
;
Amy K. Sheaffer
;
Cha
o
qun Chen
;
Min S. Lee
;
Diana Barry
;
Jay
O
.
Knipe
;
Wenying Li
;
Y
o
ng-Hae Han
;
Susan Jenkins
;
Christ
o
ph Gesenberg
;
Qi Ga
o
;
Michael W. Sinz
;
Kenneth S. Sant
o
ne
;
Tatyana Zvyaga
;
Ramkumar Rajamani
;
Herbert E. Klei
;
Richard J. C
o
l
o
nn
o
;
Dennis M. Grasela
;
Eric Hughes
;
Caly Chien
;
Stephen Adams
;
Paul C. Levesque
;
Danshi Li
;
Jial
o
ng Zhu
;
Nich
o
las A. Meanwell
;
Fi
o
na McPhee
刊名:J
o
urnal
o
f Medicinal Chemistry
出版年:2014
5.
The Disc
o
very
o
f Asunaprevir (BMS-650032), An Orally Efficaci
o
us NS3 Pr
o
tease Inhibit
o
r f
o
r the Treatment
o
f Hepatitis C Virus Infecti
o
n
作者:
Paul M. Sc
o
la
;
Li-Qiang Sun
;
Alan Xiangd
o
ng Wang
;
Jie Chen
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Anth
o
ny C
o
cuzza
;
D
o
nna M. Bilder
;
Stanley V. D鈥橝ndrea
;
Barbara Zheng
;
Piyasena Hewawasam
;
Y
o
ng Tu
;
Jacques Frib
o
rg
;
Paul Falk
;
Dennis Hernandez
;
Steven Levine
;
Cha
o
qun Chen
;
Fei Yu
;
Amy K. Sheaffer
;
Guangzhi Zhai
;
Diana Barry
;
Jay
O
.
Knipe
;
Y
o
ng-Hae Han
;
Richard Schartman
;
Maria D
o
n
o
s
o
;
Kathy M
o
sure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Andrew C. G
oo
d
;
Ramkumar Rajamani
;
Kevin Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Ga
o
;
Lucian
o
Mueller
;
Richard J. C
o
l
o
nn
o
;
Dennis M. Grasela
;
Stephen P. Adams
;
James L
o
y
;
Paul C. Levesque
;
Huabin Sun
;
H
o
ng Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jial
o
ng Zhu
;
Nich
o
las A. Meanwell
;
Fi
o
na McPhee
刊名:J
o
urnal
o
f Medicinal Chemistry
出版年:2014
6.
Cathepsin B-Labile Dipeptide Linkers f
o
r Lys
o
s
o
mal Release
o
f D
o
x
o
rubicin fr
o
m Internalizing Immun
o
c
o
njugates: M
o
del Studies
o
f Enzymatic Drug Release and Antigen-Specific In Vitr
o
Anticancer Activity
作者:
Gene M. Dub
o
wchik
;
Raym
o
nd A. Firest
o
ne
;
Linda Padilla
;
David Willner
;
Sandra J. H
o
fstead
;
Kathleen M
o
sure
;
Jay
O
.
Knipe
;
Shirley J. Lasch
;
and Pamela A. Trail
刊名:Bi
o
c
o
njugate Chemistry
出版年:2002
7.
New hydraz
o
ne derivatives
o
f Adriamycin and their immun
o
c
o
njugates - a c
o
rrelati
o
n between acid stability and cyt
o
t
o
xicity
作者:
Takushi Kanek
o
;
David Willner
;
Iv
o
M
o
nk
o
vic
;
Jay
O
.
Knipe
;
Gary R. Braslawsky
;
R
o
bert S. Greenfield
;
and D
o
latrai M. Vyas
刊名:Bi
o
c
o
njugate Chemistry
出版年:1991
8.
Methylase m
o
dels: studies
o
n general-base vs. nucle
o
philic catalysis in the intram
o
lecular alkylati
o
n
o
f phen
o
ls
作者:
Jay
O
.
Knipe
;
Peter J. Vasquez
;
and James K. C
o
ward
刊名:J
o
urnal
o
f the American Chemical S
o
ciety
出版年:1982
9.
R
o
le
o
f buffers in a methylase m
o
del reacti
o
n. General base catalysis by
o
xyani
o
ns vs. nucle
o
philic dealkylati
o
n by amines
作者:
Jay
O
.
Knipe
and James K. C
o
ward
刊名:J
o
urnal
o
f the American Chemical S
o
ciety
出版年:1979
10.
.alpha.-Deuterium is
o
t
o
pe effects and transiti
o
n-state structure in an intram
o
lecular m
o
del system f
o
r methyl-transfer enzymes
作者:
Ivan Mihel
;
Jay
O
.
Knipe
;
James K. C
o
ward
;
and Richard L. Sch
o
wen
刊名:J
o
urnal
o
f the American Chemical S
o
ciety
出版年:1979
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