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SpringerLink电子期刊(5)
Elsevier电子期刊(26)
ACS电子期刊(12)
在“
ACS电子期刊
”中,
命中:
12
条,耗时:小于0.01 秒
在所有数据库中总计命中:
43
条
1.
Discovery of Isonicotinamides as Highly Selective, Brain Penetrable, and Orally Active Glycogen Synthase Kinase-3 Inhibitors
作者:
Guanglin Luo
;
Ling Chen
;
Catherine R. Burton
;
Hong Xiao
;
Prasanna Sivaprakasam
;
Carol M. Krause
;
Yang Cao
;
Nengyin Liu
;
Jonathan Lippy
;
Wendy J. Clarke
;
Kimberly Snow
;
Joseph Raybon
;
Vinod Arora
;
Matt Pokross
;
Kevin
Kish
;
Hal A. Lewis
;
David R. Langley
;
John E. Macor
;
Gene M. Dubowchik
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery of a Potent Acyclic, Tripeptidic, Acyl Sulfonamide Inhibitor of Hepatitis C Virus NS3 Protease as a Back-up to Asunaprevir with the Potential for Once-Daily Dosing
作者:
Li-Qiang Sun
;
Eric Mull
;
Barbara Zheng
;
Stanley D’Andrea
;
Qian Zhao
;
Alan Xiangdong Wang
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Jie Chen
;
Anthony Cocuzza
;
Donna M. Bilder
;
Arvind Mathur
;
Richard Rampulla
;
Bang-Chi Chen
;
Theerthagiri Palani
;
Sivakumar Ganesan
;
Pirama Nayagam Arunachalam
;
Paul Falk
;
Steven Levine
;
Chaoqun Chen
;
Jacques Friborg
;
Fei Yu
;
Dennis Hernandez
;
Amy K. Sheaffer
;
Jay O. Knipe
;
Yong-Hae Han
;
Richard Schartman
;
Maria Donoso
;
Kathy Mosure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Ramkumar Rajamani
;
Kevin
Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Gao
;
Alicia Ng
;
Luciano Mueller
;
Dennis M. Grasela
;
Stephen Adams
;
James Loy
;
Paul C. Levesque
;
Huabin Sun
;
Hong Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jialong Zhu
;
Ying-Kai Wang
;
Hua Fang
;
Mark I. Cockett
;
Nicholas A. Meanwell
;
Fiona McPhee
;
Paul M. Scola
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Influence of Backbone Conformational Rigidity in Temperature-Sensitive Amphiphilic Supramolecular Assemblies
作者:
Krishna R. Raghupathi
;
Uma Sridhar
;
Kevin
Byrne
;
Kish
ore Raghupathi
;
S. Thayumanavan
刊名:Journal of the American Chemical Society
出版年:2015
4.
The Discovery of Asunaprevir (BMS-650032), An Orally Efficacious NS3 Protease Inhibitor for the Treatment of Hepatitis C Virus Infection
作者:
Paul M. Scola
;
Li-Qiang Sun
;
Alan Xiangdong Wang
;
Jie Chen
;
Ny Sin
;
Brian L. Venables
;
Sing-Yuen Sit
;
Yan Chen
;
Anthony Cocuzza
;
Donna M. Bilder
;
Stanley V. D鈥橝ndrea
;
Barbara Zheng
;
Piyasena Hewawasam
;
Yong Tu
;
Jacques Friborg
;
Paul Falk
;
Dennis Hernandez
;
Steven Levine
;
Chaoqun Chen
;
Fei Yu
;
Amy K. Sheaffer
;
Guangzhi Zhai
;
Diana Barry
;
Jay O. Knipe
;
Yong-Hae Han
;
Richard Schartman
;
Maria Donoso
;
Kathy Mosure
;
Michael W. Sinz
;
Tatyana Zvyaga
;
Andrew C. Good
;
Ramkumar Rajamani
;
Kevin
Kish
;
Jeffrey Tredup
;
Herbert E. Klei
;
Qi Gao
;
Luciano Mueller
;
Richard J. Colonno
;
Dennis M. Grasela
;
Stephen P. Adams
;
James Loy
;
Paul C. Levesque
;
Huabin Sun
;
Hong Shi
;
Lucy Sun
;
William Warner
;
Danshi Li
;
Jialong Zhu
;
Nicholas A. Meanwell
;
Fiona McPhee
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Structures of Kibdelomycin Bound to Staphylococcus aureus GyrB and ParE Showed a Novel U-Shaped Binding Mode
作者:
Jun Lu
;
Sangita Patel
;
Nandini Sharma
;
Stephen M. Soisson
;
Ryuta
Kish
ii
;
Masaya Takei
;
Yasumichi Fukuda
;
Kevin
J. Lumb
;
Sheo B. Singh
刊名:ACS Chemical Biology
出版年:2014
6.
Reversible Cyclic Peptide Libraries for the Discovery of Affinity Ligands
作者:
Stefano Menegatti
;
Kevin
Lawrence Ward
;
Amith Dattatray Naik
;
William Stanley
Kish
;
Robert
Kevin
Blackburn
;
Ruben Guillermo Carbonell
刊名:Analytical Chemistry
出版年:2013
7.
Optimization of Activity, Selectivity, and Liability Profiles in 5-Oxopyrrolopyridine DPP4 Inhibitors Leading to Clinical Candidate (Sa)-2-(3-(Aminomethyl)-4-(2,4-dichlorophenyl)-2-methyl-5-oxo
作者:
Pratik Devasthale
;
Ying Wang
;
Wei Wang
;
John Fevig
;
JianXin Feng
;
Aiying Wang
;
Tom Harrity
;
Don Egan
;
Nathan Morgan
;
Michael Cap
;
Aberra Fura
;
Herbert E. Klei
;
Kevin
Kish
;
Carolyn Weigelt
;
Lucy Sun
;
Paul Levesque
;
Frederic Moulin
;
Yi-Xin Li
;
Robert Zahler
;
Mark S. Kirby
;
Lawrence G. Hamann
刊名:Journal of Medicinal Chemistry
出版年:2013
8.
Synthesis and Biochemical Evaluation of Thiochromanone Thiosemicarbazone Analogues as Inhibitors of Cathepsin L
作者:
Jiangli Song
;
Lindsay M. Jones
;
G. D.
Kish
ore Kumar
;
Elizabeth S. Conner
;
Liela Bayeh
;
Gustavo E. Chavarria
;
Amanda K. Charlton-Sevcik
;
Shen-En Chen
;
David J. Chaplin
;
Mary Lynn Trawick
;
Kevin
G. Pinney
刊名:ACS Medicinal Chemistry Letters
出版年:2012
9.
Image Annotation and Database Mining to Create a Novel Screen for the Chemotype-Dependent Crystallization of HCV NS3 Protease
作者:
Herbert E. Klei
;
Kevin
Kish
;
Mark F. Russo
;
Steve J. Michalczyk
;
Matthew H. Cahn
;
Jeffrey Tredup
;
ChiehYing Chang
;
Javed Khan
;
Eric T. Baldwin
刊名:Crystal Growth & Design
出版年:2011
10.
Small Molecule Receptor Protein Tyrosine Phosphatase 纬 (RPTP纬) Ligands That Inhibit Phosphatase Activity via Perturbation of the Tryptophan鈥揚roline鈥揂spartate (WPD) Loop
作者:
Steven Sheriff
;
Brett R. Beno
;
Weixu Zhai
;
Walter A. Kostich
;
Patricia A. McDonnell
;
Kevin
Kish
;
Valentina Goldfarb
;
Mian Gao
;
Susan E. Kiefer
;
Joseph Yanchunas
;
Yanling Huang
;
Shuhao Shi
;
Shirong Zhu
;
Carolyn Dzierba
;
Joanne Bronson
;
John E. Macor
;
Kingsley K. Appiah
;
Ryan S. Westphal
;
Jonathan O鈥機onnell
;
Samuel W. Gerritz
刊名:Journal of Medicinal Chemistry
出版年:2011
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