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Elsevier电子期刊(9)
ACS电子期刊(8)
在“
ACS电子期刊
”中,
命中:
8
条,耗时:小于0.01 秒
在所有数据库中总计命中:
17
条
1.
Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quino
作者:
Felix Gonzalez-Lopez de Turiso
;
Xiaolin Hao
;
Youngsook Shin
;
Minna Bui
;
Iain D. G. Campuzano
;
Mario Cardozo
;
Michelle C. Dunn
;
Jason Duquette
;
Benjamin Fisher
;
Robert S. Foti
;
Kirk
Henne
;
Xiao He
;
Yi-Ling Hu
;
Ron C. Kelly
;
Michael G. Johnson
;
Brian S. Lucas
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Tisha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Christine Vissinga
;
Sharon Wannberg
;
Douglas A. Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery, Optimization, and in Vivo Evaluation of Benzimidazole Derivatives AM-8508 and AM-9635 as Potent and Selective PI3Kδ Inhibitors
作者:
Youngsook Shin
;
Julia Suchomel
;
Mario Cardozo
;
Jason Duquette
;
Xiao He
;
Kirk
Henne
;
Yi-Ling Hu
;
Ron C. Kelly
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Tisha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Christine Vissinga
;
Simon Wong
;
Sharon Wannberg
;
Douglas A. Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Discovery and in Vivo Evaluation of (S)-N-(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and Related PI3K未 Inhibitors for Inflammation and Autoimmune
作者:
Timothy D. Cushing
;
Xiaolin Hao
;
Youngsook Shin
;
Kristin Andrews
;
Matthew Brown
;
Mario Cardozo
;
Yi Chen
;
Jason Duquette
;
Ben Fisher
;
Felix Gonzalez-Lopez de Turiso
;
Xiao He
;
Kirk
R.
Henne
;
Yi-Ling Hu
;
Randall Hungate
;
Michael G. Johnson
;
Ron C. Kelly
;
Brian Lucas
;
John D. McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Tisha San Miguel
;
Deanna Mohn
;
Vatee Pattaropong
;
Liping H. Pettus
;
Andreas Reichelt
;
Robert M. Rzasa
;
Jennifer Seganish
;
Andrew S. Tasker
;
Robert C. Wahl
;
Sharon Wannberg
;
Douglas A. Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Dawei Zhang
;
Daniela P. Metz
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Discovery of AZD8931, an Equipotent, Reversible Inhibitor of Signaling by EGFR, HER2, and HER3 Receptors
作者:
Bernard Barlaam
;
Judith Anderton
;
Peter Ballard
;
Robert H. Bradbury
;
Laurent F. A.
Henne
quin
;
D. Mark Hickinson
;
Jason G. Kettle
;
George
Kirk
;
Teresa Klinowska
;
Christine Lambert-van der Brempt
;
Cath Trigwell
;
John Vincent
;
Donald Ogilvie
刊名:ACS Medicinal Chemistry Letters
出版年:2013
5.
Discovery and in Vivo Evaluation of Dual PI3K尾/未 Inhibitors
作者:
Felix Gonzalez-Lopez de Turiso
;
Youngsook Shin
;
Matthew Brown
;
Mario Cardozo
;
Yi Chen
;
David Fong
;
Xiaolin Hao
;
Xiao He
;
Kirk
Henne
;
Yi-Ling Hu
;
Michael G. Johnson
;
Todd Kohn
;
Julia Lohman
;
Helen J. McBride
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Kent Miner
;
Deanna Mohn
;
Vatee Pattaropong
;
Jennifer Seganish
;
Jillian L. Simard
;
Sharon Wannberg
;
Douglas A. Whittington
;
Gang Yu
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2012
6.
Bioactivation of 4-Ipomeanol by CYP4B1: Adduct Characterization and Evidence for an Enedial Intermediate
作者:
Brian R. Baer
;
Allan E. Rettie
;
and
Kirk
R.
Henne
刊名:Chemical Research in Toxicology
出版年:2005
7.
Covalent Linkage of Prosthetic Heme to CYP4 Family P450 Enzymes
作者:
Kirk
R.
Henne
;
Kent L. Kunze
;
Yi-Min Zheng
;
Peter Christmas
;
Roy J. Soberman
;
and Allan E. Rettie
刊名:Biochemistry
出版年:2001
8.
Enzymatic Determinants of the Substrate Specificity of CYP2C9: Role of B'-C Loop Residues in Providing the -Stacking Anchor Site for Wa
作者:
Robert L. Haining
;
Jeffrey P. Jones
;
Kirk
R.
Henne
;
Michael B. Fisher
;
Dennis R. Koop
;
William F. Trager
;
and Allan E. Rettie
刊名:Biochemistry
出版年:1999
1
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