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Elsevier电子期刊(14)
ACS电子期刊(11)
在“
ACS电子期刊
”中,
命中:
11
条,耗时:小于0.01 秒
在所有数据库中总计命中:
25
条
1.
5-Alkyl-2-urea-Substituted Pyridines: Identification of Efficacious Glucokinase Activators with Improved Properties
作者:
Todd J. Kohn
;
Xiaohui Du
;
SuJen Lai
;
YuMei Xiong
;
Renee Komorowski
;
Murielle Veniant
;
Zice Fu
;
Xianyun Jiao
;
Vatee Pattaropong
;
David Chow
;
Mario
Cardozo
;
Lixia Jin
;
Mario
n Conn
;
Walter E. DeWolf Jr.
;
Christopher F. Kraser
;
Ronald J. Hinklin
;
Mark L. Boys
;
Julio C. Medina
;
Jonathan Houze
;
Paul Dransfield
;
Peter Coward
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quino
作者:
Felix Gonzalez-Lopez de Turiso
;
Xiaolin Hao
;
Youngsook Shin
;
Minna Bui
;
Iain D. G. Campuzano
;
Mario
Cardozo
;
Michelle C. Dunn
;
Jason Duquette
;
Benjamin Fisher
;
Robert S. Foti
;
Kirk Henne
;
Xiao He
;
Yi-Ling Hu
;
Ron C. Kelly
;
Michael G. Johnson
;
Brian S. Lucas
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Tisha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Christine Vissinga
;
Sharon Wannberg
;
Douglas A. Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Discovery, Optimization, and in Vivo Evaluation of Benzimidazole Derivatives AM-8508 and AM-9635 as Potent and Selective PI3Kδ Inhibitors
作者:
Youngsook Shin
;
Julia Suchomel
;
Mario
Cardozo
;
Jason Duquette
;
Xiao He
;
Kirk Henne
;
Yi-Ling Hu
;
Ron C. Kelly
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Tisha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Christine Vissinga
;
Simon Wong
;
Sharon Wannberg
;
Douglas A. Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Discovery and in Vivo Evaluation of (S)-N-(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and Related PI3K未 Inhibitors for Inflammation and Autoimmune
作者:
Timothy D. Cushing
;
Xiaolin Hao
;
Youngsook Shin
;
Kristin Andrews
;
Matthew Brown
;
Mario
Cardozo
;
Yi Chen
;
Jason Duquette
;
Ben Fisher
;
Felix Gonzalez-Lopez de Turiso
;
Xiao He
;
Kirk R. Henne
;
Yi-Ling Hu
;
Randall Hungate
;
Michael G. Johnson
;
Ron C. Kelly
;
Brian Lucas
;
John D. McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Tisha San Miguel
;
Deanna Mohn
;
Vatee Pattaropong
;
Liping H. Pettus
;
Andreas Reichelt
;
Robert M. Rzasa
;
Jennifer Seganish
;
Andrew S. Tasker
;
Robert C. Wahl
;
Sharon Wannberg
;
Douglas A. Whittington
;
John Whoriskey
;
Gang Yu
;
Leeanne Zalameda
;
Dawei Zhang
;
Daniela P. Metz
刊名:Journal of Medicinal Chemistry
出版年:2015
5.
Absorption and Fluorescence Spectra of Poly(p-phenylenevinylene) (PPV) Oligomers: An ab Initio Simulation
作者:
Thiago M.
Cardozo
;
Ad茅lia J. A. Aquino
;
Mario
Barbatti
;
Itamar Borges
;
Jr.
;
Hans Lischka
刊名:Journal of Physical Chemistry A
出版年:2015
6.
Discovery and in Vivo Evaluation of Dual PI3K尾/未 Inhibitors
作者:
Felix Gonzalez-Lopez de Turiso
;
Youngsook Shin
;
Matthew Brown
;
Mario
Cardozo
;
Yi Chen
;
David Fong
;
Xiaolin Hao
;
Xiao He
;
Kirk Henne
;
Yi-Ling Hu
;
Michael G. Johnson
;
Todd Kohn
;
Julia Lohman
;
Helen J. McBride
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Kent Miner
;
Deanna Mohn
;
Vatee Pattaropong
;
Jennifer Seganish
;
Jillian L. Simard
;
Sharon Wannberg
;
Douglas A. Whittington
;
Gang Yu
;
Timothy D. Cushing
刊名:Journal of Medicinal Chemistry
出版年:2012
7.
Structure-Guided Design, Synthesis, and Evaluation of Guanine-Derived Inhibitors of the eIF4E mRNA鈥揅ap Interaction
作者:
Xiaoqi Chen
;
David J. Kopecky
;
Jeff Mihalic
;
Shawn Jeffries
;
Xiaoshan Min
;
Julie Heath
;
Jeff Deignan
;
SuJen Lai
;
Zice Fu
;
Cristiano Guimaraes
;
Shanling Shen
;
Shyun Li
;
Sheree Johnstone
;
Stephen Thibault
;
Haoda Xu
;
Mario
Cardozo
;
Wang Shen
;
Nigel Walker
;
Frank Kayser
;
Zhulun Wang
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
Thermodynamic Analysis of mRNA Cap Binding by the Human Initiation Factor eIF4E via Free Energy Perturbations
作者:
Cristiano R. W. Guimares
;
David J. Kopecky
;
Jeff Mihalic
;
Shanling Shen
;
Shawn Jeffries
;
Stephen T. Thibault
;
Xiaoqi Chen
;
Nigel Walker
;
Mario
Cardozo
刊名:Journal of the American Chemical Society
出版年:2009
9.
MM-GB/SA Rescoring of Docking Poses in Structure-Based Lead Optimization
作者:
Cristiano R. W. Guimarã
;
es
;
Mario
Cardozo
刊名:Journal of Chemical Information and Modeling
出版年:2008
10.
Significance Analysis and Multiple Pharmacophore Models for Differentiating P-Glycoprotein Substrates
作者:
Wu-Xiong Li
;
Leping Li
;
John Eksterowicz
;
Xuefeng Bruce Ling
;
Mario
Cardozo
刊名:Journal of Chemical Information and Modeling
出版年:2007
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