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SpringerLink电子期刊(15)
Elsevier电子期刊(55)
ACS电子期刊(8)
在“
ACS电子期刊
”中,
命中:
8
条,耗时:0.0449412 秒
在所有数据库中总计命中:
78
条
1.
S
ulfonamide
s
a
s
Selective NaV1.7 Inhibitor
s
: Optimizing Potency and Pharmacokinetic
s
to Enable in Vivo Target Engagement
作者:
I
s
aac E. Marx
;
Thoma
s
A. Dineen
;
Je
ss
ica Able
;
Chri
s
tiane Bode
;
Howard Bregman
;
Margaret Chu-Moyer
;
Erin F. DiMauro
;
Bingfan Du
;
Robert
S
.
Foti
;
Robert
T. Fremeau Jr.
;
Hua Gao
;
Hakan Gunaydin
;
Brian E. Hall
;
Liyue Huang
;
Thoma
s
Kornecook
;
Charle
s
R. Kreiman
;
Daniel
S
. La
;
Jo
s
eph Ligutti
;
Min-Hwa Ja
s
mine Lin
;
Dong Liu
;
Jeff
S
. McDermott
;
Bryan D. Moyer
;
Emily A. Peter
s
on
;
Jonathan T.
Roberts
;
Paul Ro
s
e
;
Jean Wang
;
Beth D. Youngblood
;
Violeta Yu
;
Matthew M. Wei
ss
刊名:AC
S
Medicinal Chemi
s
try Letter
s
出版年:2016
2.
Di
s
covery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitor
s
2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quino
作者:
Felix Gonzalez-Lopez de Turi
s
o
;
Xiaolin Hao
;
Young
s
ook Shin
;
Minna Bui
;
Iain D. G. Campuzano
;
Mario Cardozo
;
Michelle C. Dunn
;
Ja
s
on Duquette
;
Benjamin Fi
s
her
;
Robert
S
.
Foti
;
Kirk Henne
;
Xiao He
;
Yi-Ling Hu
;
Ron C. Kelly
;
Michael G. John
s
on
;
Brian
S
. Luca
s
;
John McCarter
;
Lawrence R. McGee
;
Julio C. Medina
;
Daniela Metz
;
Ti
s
ha San Miguel
;
Deanna Mohn
;
Thuy Tran
;
Chri
s
tine Vi
ss
inga
;
S
haron Wannberg
;
Dougla
s
A. Whittington
;
John Whori
s
key
;
Gang Yu
;
Leeanne Zalameda
;
Xuxia Zhang
;
Timothy D. Cu
s
hing
刊名:Journal of Medicinal Chemi
s
try
出版年:2016
3.
Application of a Parallel
S
ynthetic Strategy in the Di
s
covery of Biaryl Acyl Sulfonamide
s
a
s
Efficient and Selective NaV1.7 Inhibitor
s
作者:
Erin F. DiMauro
;
S
tephen Altmann
;
Loren M. Berry
;
Howard Bregman
;
Naga
s
ree Chakka
;
Margaret Chu-Moyer
;
Elma Feric Bojic
;
Robert
S
.
Foti
;
Robert
Fremeau
;
Hua Gao
;
Hakan Gunaydin
;
Angel Guzman-Perez
;
Brian E. Hall
;
Hongbing Huang
;
Michael Jaro
s
h
;
Thoma
s
Kornecook
;
Jo
s
ie Lee
;
Jo
s
eph Ligutti
;
Dong Liu
;
Bryan D. Moyer
;
Daniel Ortuno
;
Paul E. Ro
s
e
;
Laurie B.
S
chenkel
;
Kri
s
tin Taborn
;
Jean Wang
;
Yan Wang
;
Violeta Yu
;
Matthew M. Wei
ss
刊名:Journal of Medicinal Chemi
s
try
出版年:2016
4.
Catalytic ver
s
u
s
Inhibitory Promi
s
cuity in Cytochrome P450
s
: Implication
s
for Evolution of New Function
作者:
Robert
S
.
Foti
;
Mathew Honaker
;
Abhinav Nath
;
Jo
s
h T. Pear
s
on
;
Brian Buttrick
;
Nina I
s
oherranen
;
William M. Atkin
s
刊名:Biochemi
s
try
出版年:2011
5.
Ligand-Ba
s
ed De
s
ign of a Potent and Selective Inhibitor of Cytochrome P450 2C19
作者:
Robert
S
.
Foti
;
Dan A. Rock
;
Xiaogang Han
;
Robert
A. Flower
s
;
II
;
Larry C. Wienker
s
;
Jan L. Wahl
s
trom
刊名:Journal of Medicinal Chemi
s
try
出版年:2012
6.
4-Hydroxy-1,2,5-oxadiazol-3-yl Moiety a
s
Bioi
s
o
s
ter of the Carboxy Function. Synthe
s
i
s
, Ionization Con
s
tant
s
, and Molecular Pharmacological Characterization at Ionotropic Glutamate Receptor
s
of Compou
作者:
Marco L. Lolli
;
Cecilia Giordano
;
Darryl
S
. Pickering
;
Barbara Rolando
;
Ka
s
per B. Han
s
en
;
Antonio
Foti
;
Alberto Contrera
s
-Sanz
;
Ahmad Amir
;
Robert
a Fruttero
;
Alberto Ga
s
co
;
Birgitte Niel
s
en
;
Tommy N. J
刊名:Journal of Medicinal Chemi
s
try
出版年:2010
7.
Differential Time-Dependent Inactivation of P450 3A4 and P450 3A5 by Raloxifene: A Key Role for C239 in Quenching Reactive Intermediate
s
作者:
Jo
s
h T. Pear
s
on
;
Jan L. Wahl
s
trom
;
Le
s
lie J. Dickmann
;
S
anto
s
h Kumar
;
Jame
s
R. Halpert
;
Larry C. Wienker
s
;
Robert
S
.
Foti
;
Dan A. Rock
刊名:Chemical Re
s
earch in Toxicology
出版年:2007
8.
N
s
LTP1 and N
s
LTP2 I
s
oform
s
in Soft Wheat (Triticum ae
s
tivum Cv. Centauro) and Farro (Triticum dicoccon Schrank) Bran
作者:
Antonella Capocchi
;
Debora Fontanini
;
Vera Muccilli
;
Vincenzo Cun
s
olo
;
Franco
S
aviozzi
;
Ro
s
aria Saletti
;
Robert
o Lorenzi
;
S
alvatore
Foti
;
and Luciano Galle
s
chi
刊名:Journal of Agricultural and Food Chemi
s
try
出版年:2005
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