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Wiley电子期刊(16)	NATURE电子期刊(11)	ACS电子期刊(247)
SpringerLink电子期刊(368)	Elsevier电子期刊(1333)

在“Elsevier电子期刊”中，命中：1,333条，耗时：0.0269876 秒

在所有数据库中总计命中：1,975条

1.Towards the development of activity-based probes for detection of lysine-specific demethylase-1 activity

作者：Maria E. Ourailidou^a ; Alessia Lenoci^b ; Clemens Zwergel^b ; Dante Rotili^b ; Antonello Mai^b ; ^c ; ^{antonello.mai@uniroma1.it} ; Frank J. Dekker^a ; ^{f.j.dekker@rug.nl}

关键词：Lysine demethylation ; Tumorigenesis ; Tranylcypromine ; Irreversible inhibition ; Enzyme labeling

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

2.mTOR Inhibition Mitigates Molecular and Biochemical Alterations of Vigabatrin-Induced Visual Field Toxicity in Mice

作者：Kara R. Vogel ; PhD^a ; Garrett R. Ainslie ; PhD^a ; Michelle A. Schmidt ; MS^b ; Jonathan P. Wisor ; PhD^b ; K. Michael Gibson ; PhD^a ; ^{mike.gibson@wsu.edu}

关键词：vigabatrin ; GABA ; mTOR ; gene expression ; visual evoked potentials ; visual field loss ; ARPE19 cells ; epilepsy

刊名：Pediatric Neurology

出版年：2017

3.Irreversible electroporation inhibits pro-cancer inflammatory signaling in triple negative breast cancer cells

作者：Ishan Goswami^aAuthor Vitae ; Sheryl Coutermarsh-Ott^cAuthor Vitae ; Ryan G. Morrison^bAuthor Vitae ; Irving C. Allen^cAuthor Vitae ; Rafael V. Davalos^a ; ^b ; ^dAuthor Vitae ; Scott S. Verbridge^b ; ^d ; ^{sverb@vt.edu" class="auth_mail" title="E-mail the corresponding author}Author Vitae ; Lissett R. Bickford^a ; ^b ; ^dAuthor Vitae

关键词：Electroporation ; Triple negative breast cancer ; Thymic stromal lymphopoietin (TSLP) ; Immunotherapy

刊名：Bioelectrochemistry

出版年：2017

4.Inhibiting medial septal cholinergic neurons with DREADD alleviated anxiety-like behaviors in mice

作者：Yu Zhang^a ; Ying-Ying Jiang^a ; Shan Shao^a ; Chan Zhang^a ; Feng-Yu Liu^a ; You Wan^a ; ^b ; ^c ; Ming Yi^a ; ^{mingyi@bjmu.edu.cn}

关键词：ChAT ; choline acetyltransferase ; CNO ; clozapine N-oxide ; DREADD ; designer receptors exclusively activated by designer drugs ; EPM ; elevated plus-maze ; MB ; marble burying ; MS ; medial septum ; NSF ; novelty-suppressed feeding ; OF ; open field ; PFA ; paraformaldehyde ; PV ; parvalbumin ; SAP ; 192 IgG-saporin

刊名：Neuroscience Letters

出版年：2017

5.The performance of activated sludge exposed to arsanilic acid and amprolium hydrochloride in sequencing batch reactors

作者：Kui Chen^a ; Feng Ji^b ; Shoujun Yuan^a ; ^d ; Wentao Hao^c ; Wei Wang^a ; ^d ; ^{dwhit@126.com} ; Zhen-Hu Hu^a ; ^d ; ^{zhhu@hfut.edu.cn}

关键词：Activated sludge ; Arsanilic acid (ASA) ; Amprolium hydrochloride (AMP) ; Nutrient removal

刊名：International Biodeterioration & Biodegradation

出版年：2017

6.Proteasome inhibition by new dual warhead containing peptido vinyl sulfonyl fluorides

作者：Arwin J. Brouwer^a ; ^&dagger ; ; Natalia Herrero Á ; lvarez^b ; ^&dagger ; ; Adriano Ciaffoni^a ; Helmus van de Langemheen^b ; Rob M.J. Liskamp^a ; ^b ; ^{r.m.j.liskamp@uu.nl" class="auth_mail" title="E-mail the corresponding author} ; ^{Robert.liskamp@glasgow.ac.uk" class="auth_mail" title="E-mail the corresponding author}

关键词：Drug design ; Peptido vinyl sulfonyl fluoride ; Proteasome ; Irreversible inhibition ; Dual warhead

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

7.Synthesis, structural characterization, docking, lipophilicity and cytotoxicity of 1-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-3-alkyl carbamates, novel acetylcholinesterase and butyrylcholinesterase pseudo-irreversible inhibitors

作者：Vladimí ; r Pejchal^a ; ^{vladimir.pejchal@upce.cz" class="auth_mail" title="E-mail the corresponding author} ; &Scaron ; á ; rka &Scaron ; těpá ; nková ; ^b ; Marcela Pejchalová ; ^b ; Karel Krá ; lovec^b ; Radim Havelek^b ; Zdeňka Růžičková ; ^c ; Haresh Ajani^d ; ^e ; Rabindranath Lo^d ; Martin Lep&scaron ; í ; k^d

关键词：Halogenated benzothiazole ; Carbamates ; Acetylcholinesterase ; Butyrylcholinesterase inhibition ; Pseudo-irreversible mechanism ; Covalent docking

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

作者：Le Min ^{lmin@bwh.harvard.edu}

关键词：Cancer ; Hypophysitis ; Immune checkpoint inhibition ; Immune-related adverse events ; Thyroiditis

刊名：Genes & Diseases

出版年：2016

9.Multiple modes of inhibition of human cytochrome P450 2J2 by dronedarone, amiodarone and their active metabolites

作者：Aneesh Karkhanis^a ; Hui Yuan Lam^a ; Gopalakrishnan Venkatesan^a ; Siew Kwan Koh^b ; Christina Li Lin Chai^a ; Lei Zhou^b ; Yanjun Hong^a ; Pipin Kojodjojo^c ; Eric Chun Yong Chan^a ; ^{phaccye@nus.edu.sg" class="auth_mail" title="E-mail the corresponding author}

关键词：AA ; arachidonic acid ; ACN ; acetonitrile ; AF ; atrial fibrillation ; CYP2D6 ; cytochrome P450 2D6 ; CYP2J2 ; cytochrome P450 2J2 ; CYP3A4 ; cytochrome P450 3A4 ; CYP3A5 ; cytochrome P450 3A5 ; DDI ; drug&ndash ; drug interaction ; EET ; epoxyeicosatrienoic acid ; GSH ; glutathione ; k ; intrinsic elimination rate constant ; Ki ; reversible inhibition constant ; KI ; inactivator concentration at half-maximum inactivation rate constant ; kinact ; maximum inactivation rate constant ; Km ; Michaelis&ndash ; Menten constant ; Kobs

刊名：Biochemical Pharmacology

出版年：2016

10.Design, synthesis and biological evaluation of N-methyl-N-[(1,2,3-triazol-4-yl)alkyl]propargylamines as novel monoamine oxidase B inhibitors

作者：Ornella Di Pietro^a ; Nelson Alencar^b ; Gerard Esteban^c ; Elisabet Viayna^a ; Natalia Szałaj^a ; Javier Vá ; zquez^b ; Jordi Juá ; rez-Jimé ; nez^b ; Irene Sola^a ; Belé ; n Pé ; rez^d ; Montse Solé ; ^c ; Mercedes Unzeta^c ; Diego Muñ ; oz-Torrero^a ; ^{dmunoztorrero@ub.edu" class="auth_mail" title="E-mail the corresponding author} ; F. Javier Luque^b ; ^{fjluque@ub.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：Click-chemistry ; Monoamine oxidase B ; Alzheimer&rsquo ; s disease ; Irreversible inhibition

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

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