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内部出版物
SpringerLink电子期刊(7)
Elsevier电子期刊(15)
ACS电子期刊(11)
在“
Elsevier电子期刊
”中,
命中:
15
条,耗时:小于0.01 秒
在所有数据库中总计命中:
33
条
1.
Novel phenylalanine derived diamides as Factor XIa inhibitors
作者:
Leon M. Smith II
;
leon.smith@bms.com" class="auth_mail" title="E-mail the corresponding author
;
Michael J. Orwat
;
Zilun Hu
;
Wei Han
;
Cailan Wang
;
Karen A. Rossi
;
Paul J. Gilligan
;
Kumar B. Pabbisetty
;
Honey Osuna
;
James R. Corte
;
Alan R. Rendina
;
Joseph M. Luettgen
;
Pancras
C.
Wong
;
Ranga Narayanan
;
Timothy W. Harper
;
Jeffrey M. Bozarth
;
Earl J. Crain
;
Anzhi Wei
;
Vidhyashankar Ramamurthy
;
Paul E. Morin
;
Baomin Xin
;
Joanna Zheng
;
Dietmar A. Seiffert
;
Mimi L. Quan
;
Patrick Y.S. Lam
;
Ruth R. Wexler
;
Donald J.P. Pinto
关键词:
Factor XIa
;
FXIa
;
Anticoagulant
;
Thrombosis
;
Serine protease
;
aPTT
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
Synthesis and P1′ SAR exploration of potent macrocyclic tissue factor-factor VIIa inhibitors
作者:
Vladimir (Uladzimir) Ladziata
;
vladimir.ladziata@bms.com" class="auth_mail" title="E-mail the corresponding author
;
Peter W. Glunz
;
Yan Zou
&dagger
;
;
Xiaojun Zhang
;
Wen Jiang
;
Swanee Jacutin-Porte
;
Daniel L. Cheney
;
Anzhi Wei
;
Joseph M. Luettgen
;
Timothy M. Harper
;
Pancras
C.
Wong
;
Dietmar Seiffert
;
Ruth R. Wexler
;
E. Scott Priestley
关键词:
Thrombosis
;
Anticoagulant
;
Factor VIIa-TF inhibitor
;
Macrocycle
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
3.
097 - Differential Cardiac Effects of an AT1R Biased Ligand, AT1R Antagonist and ACE Inhibitor in Mouse Models of Post-Myocardial Infarction Heart Failure
作者:
Xiuying Ma
;
Shahid Tannu
;
John Allocco
;
Dike Qiu
;
Marisa Flaim
;
Earl Crain
;
Jeffrey Bostwick
;
Patricia Smith
;
Xue-Qing Chen
;
William Schumacher
;
Brian J. Arey
;
Pancras
Wong
刊名:Journal of Cardiac Failure
出版年:2016
4.
Discovery of diarylurea P2Y
1
antagonists with improved aqueous solubility
作者:
Tammy C. Wang
;
Jennifer X. Qiao
;
jennifer.qiao@bms.com
;
Charles G. Clark
;
Ji Jua
;
Laura A. Price
;
Qimin Wu
;
Ming Chang
;
Joanna Zheng
;
Christine S. Huang
;
Gerry Everlof
;
William A. Schumacher
;
Pancras
C.
Wong
;
Dietmar A. Seiffert
;
Anne B. Stewart
;
Jeffrey S. Bostwick
;
Earl J. Crain
;
Carol A. Watson
;
Robert Rehfuss
;
Ruth R. Wexler
;
Patrick Y.S. Lam
&dagger
;
关键词:
P2Y1 antagonists
;
Diarylurea
;
Structure&ndash
;
activity relationship (SAR)
;
Aqueous solubility
;
In vivo efficacy/bleeding model
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
5.
Design and synthesis of bicyclic pyrazinone and pyrimidinone amides as potent TF-FVIIa inhibitors
作者:
Xiaojun Zhang
;
xiaojun.zhang@bms.com
;
Peter W. Glunz
;
Wen Jiang
;
Aaron Schmitt
;
Makenzie Newman
;
Frank A. Barbera
;
Jeffery M. Bozarth
;
Alan R. Rendina
;
Anzhi Wei
;
Xiao Wen
;
Karen A. Rossi
;
Joseph M. Luettgen
;
Pancras
C.
Wong
;
Robert M. Knabb
;
Ruth R. Wexler
;
E. Scott Priestley
关键词:
TF&ndash
;
FVIIa inhibitor
;
Bicyclic pyrazinone
;
Bicyclic pyrimidinone
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
6.
Nonbenzamidine acylsulfonamide tissue factor-factor VIIa inhibitors
作者:
Peter W. Glunz
;
Xiaojun Zhang
;
Yan Zou
;
Indawati Delucca
;
Alex
;
ra H. Nirschl
;
Xuhong Cheng
;
Carolyn A. Weigelt
;
Daniel L. Cheney
;
Anzhi Wei
;
Rushith Anumula
;
Joseph M. Luettgen
;
Alan R. Rendina
;
Mark Harpel
;
Gang Luo
;
Robert Knabb
;
Pancras
C.
Wong
;
Ruth R. Wexler
;
E. Scott Priestley
关键词:
Factor VIIa
;
Tissue factor
;
TF-FVIIa inhibitor
;
Serine protease inhibitors
;
Structure-based design
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
7.
Highly efficacious factor Xa inhibitors containing α-substituted phenylcycloalkyl P4 moieties
作者:
Jennifer X. Qiao
;
Sarah R. King
;
Kan He
;
Pancras
C.
Wong
;
Alan R. Rendina
;
Joseph M. Luettgen
;
Baomin Xin
;
Robert M. Knabb
;
Ruth R. Wexler
;
Patrick Y.S. Lam
关键词:
Factor Xa inhibitors
;
α
;
-Substituted phenylcyclopropyls
;
SAR
;
Pharmacokinetic
;
Rabbit arterio-venous shunt
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
8.
Structure–activity relationships of anthranilamide-based factor Xa inhibitors containing piperidinone and pyridinone P4 moieties
作者:
James R. Corte
;
Tianan Fang
;
Donald J.P. Pinto
;
Wei Han
;
Zilun Hu
;
Xiang-Jun Jiang
;
Yun-Long Li
;
Jolicia F. Gauuan
;
Mark Hadden
;
Darren Orton
;
Alan R. Rendina
;
Joseph M. Luettgen
;
Pancras
C.
Wong
;
Kan
关键词:
Factor Xa
;
Anthranilamide
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
9.
Prediction of the therapeutic index of marketed anti-coagulants and anti-platelet agents by guinea pig models of thrombosis and hemostasis
作者:
J. Eileen Bird
;
Mary R. Giancarli
;
Nick Allegretto
;
Frank Barbera
;
Pancras
Wong
;
William A. Schumacher
;
Martin L. Ogletree
;
Dietmar Seiffert
关键词:
Argatroban
;
Aspirin
;
Clopidogrel
;
Hirudin
;
Tirofiban
刊名:Thrombosis Research
出版年:2008
10.
Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residues
作者:
Jennifer X. Qiao
;
Xuhong Cheng
;
Joanne M. Smallheer
;
Robert A. Galemmo
;
Spencer Drummond
;
Donald J.P. Pinto
;
Daniel L. Cheney
;
Kan He
;
Pancras
C.
Wong
;
Joseph M. Luettgen
;
et al.
关键词:
Factor Xa inhibitors
;
Pyrazole-based
;
SAR
;
N
-Arylpiperidine
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2007
1
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