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NATURE电子期刊(3)
Elsevier电子期刊(14)
ACS电子期刊(10)
在“
Elsevier电子期刊
”中,
命中:
14
条,耗时:0.0149926 秒
在所有数据库中总计命中:
27
条
1.
Chemerin-induced arterial contraction is G
i
- and calcium-dependent
作者:
David J. Ferland
;
ferlandd@msu.edu
;
Emma S. Darios
;
Richard R. Neubig
;
Benita Sjö
;
gren
;
Nguyen Truong
;
Rosa Torres
;
Thomas
S.
Dexheimer
;
Janice M. Thompson
;
Stephanie W. Watts
关键词:
Akt
;
protein kinase B
;
ANG II
;
angiotensin II
;
CaM
;
calmodulin
;
CCRL2
;
chemokine (CC motif) receptor-like 2
;
CMKLR1
;
chemokine-like receptor 1
;
Erk MAPK
;
extracellular signal-regulated kinase mitogen activated protein kinase
;
GAP
;
GTPase activating protein
;
GEF
;
guanine nucleotide exchange factor
;
GPR1
;
G protein-coupled receptor 1
;
MLC
;
myosin light-chain
;
MLCK
;
myosin light-chain kinase
;
MLCP
;
myosin light-chain phosphatase
;
PD098059
;
2-(2-amino-3-methoxyphenyl)-4H-chromen-4-one
;
PE
;
phenyleph
刊名:Vascular Pharmacology
出版年:2017
2.
Magnetic Resonance Imaging Zygapophyseal Joint Space Changes (Gapping) in Low Back Pain Patients Following Spinal Manipulation and Side-Posture Positioning: A Randomized Controlled Mechanisms Trial With Blinding
作者:
Gregory D. Cramer
;
Jerrilyn Cambron
;
Joe A. Cantu
;
Jennifer M.
Dexheimer
;
Judith D. Pocius
;
Douglas Gregerson
;
Michael Fergus
;
Ray McKinnis
;
Thomas
J. Grieve
关键词:
Manipulation
;
Spinal
;
Zygapophyseal Joint
;
Chiropractic
;
Low Back Pain
;
Lumbar Vertebrae
刊名:Journal of Manipulative and Physiological Therapeutics
出版年:2013
3.
Synthesis and SAR studies of 5-(pyridin-4-yl)-1,3,4-thiadiazol-2-amine derivatives as potent inhibitors of Bloom helicase
作者:
Andrew S. Rosenthal
;
Thomas
S.
Dexheimer
;
Opher Gileadi
;
Giang H. Nguyen
;
Wai Kit Chu
;
Ian D. Hickson
;
Ajit Jadhav
;
Anton Simeonov
;
David J. Maloney
关键词:
BLM
;
Bloom helicase
;
SAR
;
structure activity relationship
;
HTS
;
high throughput screen
;
ADME
;
absorption
;
distribution
;
metabolism and excretion
;
MLM
;
mouse liver microsomes
;
NADPH
;
nicotinamide adenine dinucleotide phosphate
;
PBS
;
phosphate buffered sali
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
4.
A Small Molecule Inhibitor of the BLM Helicase Modulates Chromosome Stability in Human Cells
作者:
Giang Huong Nguyen
1
;
2
;
7
;
Thomas
S.
Dexheimer
3
;
7
;
Andrew S. Rosenthal
3
;
Wai Kit Chu
4
;
Dharmendra Kumar Singh
6
;
Georgina Mosedale
1
;
Csaná
;
d Z. Bachrati
1
;
Lena Schultz
3
;
Masaaki Sakurai
3
;
Pavel Savitsky
5
;
Mika Abu
1
;
Peter J. McHugh
1
;
Vilhelm A. Bohr
6
;
Curtis C. Harris
2
;
Ajit Jadhav
3
;
Opher Gileadi
5
;
David J. Maloney
3
;
Anton Simeonov
3
;
asimeono@mail.nih.gov
;
Ian D. Hickson
1
;
4
;
iandh@sund.ku.dk
刊名:Chemistry & Biology
出版年:2013
5.
Shoe Orthotics for the Treatment of Chronic Low Back Pain: A Randomized Controlled Pilot Study
作者:
Jerrilyn A. Cambron DC
;
PhD
a
;
jcambron@nuhs.edu"" rel=""nofollow
;
Manuel Duarte DC
b
;
Jennifer
Dexheimer
BS
;
LMT
c
;
Thomas
Solecki DC
d
关键词:
Orthotic Devices
;
Shoes
;
Low Back Pain
;
Chiropractic
;
Biomechanics
刊名:Journal of Manipulative and Physiological Therapeutics
出版年:2011
6.
Selective and Cell-Active Inhibitors of the USP1/ UAF1 Deubiquitinase Complex Reverse Cisplatin Resistance in Non-small Cell Lung Cancer Cells
作者:
Junjun Chen
1
;
Thomas
;
S.
Dexheimer
2
;
Yongxing Ai
1
;
Qin Liang
1
;
Mark
;
A. Villamil
1
;
James Inglese
2
;
David
;
J. Maloney
2
;
Ajit Jadhav
2
;
Anton Simeonov
2
;
;
asimeono@mail.nih.gov
;
Zhihao Zhuang
1
;
;
zzhuang@udel.edu
刊名:Chemistry & Biology
出版年:2011
7.
Virtual screening using ligand-based pharmacophores for inhibitors of human tyrosyl-DNA phospodiesterase (hTdp1)
作者:
Iwona E. Weidlich
;
Thomas
S.
Dexheimer
;
Christophe March
;
Smitha Antony
;
Yves Pommier
;
Marc C. Nicklaus
关键词:
Human tyrosyl-DNA phosphodiesterase
;
Tdp1
;
Inhibitors
;
Small molecule docking
;
Drug design
;
Virtual screening
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
8.
The structure–activity relationships of A-ring-substituted aromathecin topoisomerase I inhibitors strongly support a camptothecin-like binding mode
作者:
Maris A. Cinelli
;
Andrew E. Morrell
;
Thomas
S.
Dexheimer
;
Keli Agama
;
Surbhi Agrawal
;
Yves Pommier
;
Mark Cushman
关键词:
Topoisomerase 1
;
Aromathecins
;
Anticancer
;
Camptothecin-like
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
9.
Inhibitors of human tyrosyl-DNA phospodiesterase (hTdp1) developed by virtual screening using ligand-based pharmacophores
作者:
Iwona E. Weidlich
;
Thomas
Dexheimer
;
Christophe March
;
Smitha Antony
;
Yves Pommier
;
Marc C. Nicklaus
关键词:
Human tyrosyl-DNA phosphodiesterase
;
Tdp1
;
Inhibitors
;
Small molecule docking
;
Drug design
;
Virtual screening
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
10.
Expression profiling identifies epoxy anthraquinone derivative as a DNA topoisomerase inhibitor
作者:
Jinesh Gheeya
;
Peter Johansson
;
Qing-Rong Chen
;
Thomas
Dexheimer
;
Belhu Metaferia
;
Young K. Song
;
Jun S. Wei
;
Jianbin He
;
Yves Pommier
;
Javed Khan
关键词:
Neuroblastoma
;
Anti-cancer drug
;
Microarray
;
cMAP
;
Topoisomerase
;
EAD
刊名:Cancer Letters
出版年:2010
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