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Elsevier电子期刊(9)
ACS电子期刊(4)
在“
Elsevier电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
13
条
1.
Identification and SAR of novel pyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)
作者:
Giovanna
Pescatore
;
Danila Branca
;
Fabrizio Fiore
;
Olaf Kinzel
;
Laura Llauger Bufi
;
Ester Muraglia
;
Federica Orvieto
;
Michael Rowley
;
Carlo Toniatti
;
Caterina Torrisi
;
Philip Jones
关键词:
Pyrrolo[1
;
2-
a
]pyrazin-1(2
H
)-one
;
Poly(ADP-ribose) polymerase
;
PARP-1
;
Oncology
;
Selectivity
;
BRCA1
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
2.
A novel base-mediated intramolecular hydroamination to build fused heteroaryl pyrazinones
作者:
Laura Llauger
;
Costanza Bergami
;
Olaf D. Kinzel
;
Samuele Lillini
;
Giovanna
Pescatore
;
Caterina Torrisi
;
Philip Jones
关键词:
Intramolecular hydroamination
;
Pyrrolopyrazinones
;
Fused-heteroaryl pyrazinones
;
DBU-mediated cyclisation
;
Isomerisation
刊名:Tetrahedron Letters
出版年:2009
3.
Dihydroxy-pyrimidine and N
作者:
Emanuela Nizi
;
Maria Vittoria Orsale
;
Benedetta Crescenzi
;
Giovanna
Pescatore
;
Ester Muraglia
;
Anna Alfieri
;
Cristina Gardelli
;
Sté
;
phane A.H. Spieser
;
Vincenzo Summa
关键词:
HIV-1 integrase
;
Pyrimidines
;
N
-Methylpyrimidones
;
PAMPA
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
4.
Optimization of a series of potent and selective ketone histone deacetylase inhibitors
作者:
Giovanna
Pescatore
;
Olaf Kinzel
;
Barbara Attenni
;
Ottavia Cecchetti
;
Fabrizio Fiore
;
Massimiliano Fonsi
;
Michael Rowley
;
Carsten Schultz-Fademrecht
;
Sergio Serafini
;
Christian Steinkü
;
hler
;
Philip
关键词:
HDAC inhibitors
;
Alkyl ketone
;
Zinc binding group
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
5.
The synthesis of tetrahydropyridopyrimidones as a new scaffold for HIV-1 integrase inhibitors
作者:
Olaf D. Kinzel
;
Edith Monteagudo
;
Ester Muraglia
;
Federica Orvieto
;
Giovanna
Pescatore
;
Maria del Rosario Rico Ferreira
;
Michael Rowley
;
Vincenzo Summa
关键词:
Tetrahydropyridopyrimidone
;
Integrase inhibitor
;
1
2 ;
4-Oxadiazoline
;
Amidoxime
刊名:Tetrahedron Letters
出版年:2007
6.
Tetrazole thioacetanilides: Potent non-nucleoside inhibitors of WT HIV reverse transcriptase and its K103N mutant
作者:
Ester Muraglia
;
Olaf D. Kinzel
;
Ralph Laufer
;
Michael D. Miller
;
Gregory Moyer
;
Vandna Munshi
;
Federica Orvieto
;
Maria Cecilia Palumbi
;
Giovanna
Pescatore
;
Michael Rowley
et al.
关键词:
HIV
;
Non-nucleoside reverse transcriptase inhibitors
;
Tetrazole thioacetanilides
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2006
7.
New stereoselective synthesis of the peptidic aminopeptidase inhibitors bestatin, phebestin and probestin
作者:
Righi
;
Giuliana
;
D'Achille
;
Claudia
;
Pescatore
;
Giovanna
;
Bonini
;
Carlo
关键词:
asymmetric synthesis
;
α
;
β
;
-epoxy esters
;
aminopeptidase inhibitors
刊名:Tetrahedron Letters
出版年:2003
8.
A study on the chelation control in the regioselective opening of 2,3-bifunctionalized epoxides
作者:
Righi
;
Giuliana
;
Pescatore
;
Giovanna
;
Bonadies
;
Francesco
;
Bonini
;
Carlo
关键词:
bifunctionalized epoxides
;
chelation control
;
regioselective opening
刊名:Tetrahedron
出版年:2001
9.
Holocene Coastal Environments near Pompeii before the A.D. 79 Eruption of Mount Vesuvius, Italy
作者:
Pescatore
;
Tullio
;
Senatore
;
Maria Rosaria
;
Capretto
;
Giovanna
;
Lerro
;
Gaia
刊名:Quaternary Research
出版年:2001
1
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