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Wiley电子期刊(8)
NATURE电子期刊(2)
ACS电子期刊(76)
SpringerLink电子期刊(147)
Elsevier电子期刊(465)
在“
Elsevier电子期刊
”中,
命中:
465
条,耗时:0.0149909 秒
在所有数据库中总计命中:
698
条
1.
Synthesis, structure and properties of N-aminosaccharin - A selective
inhibitor
of human
carbonic
anhydrase
I
作者:
Mikhail A. Kuznetsov
a
;
m.kuznetsov@spbu.ru
;
Aleksandr N. Shestakov
a
;
Mikhail Zibinsky
a
;
Mikhail Krasavin
a
;
Claudiu T. Supuran
b
;
Stanislav Kalinin
a
;
Muhammet Tanç
;
b
关键词:
N-Aminosaccharin
;
N-Amination
;
hCA I
inhibitor
;
Oxidative aminoaziridination
;
Ligand efficiency
刊名:Tetrahedron Letters
出版年:2017
2.
Sulfonamide inhibition profile of the γ-
carbonic
anhydrase
identified in the genome of the pathogenic bacterium Burkholderia pseudomallei the etiological agent responsible of melioidosis
作者:
Sonia Del Prete
a
;
Daniela Vullo
b
;
Pietro Di Fonzo
a
;
Sameh M. Osman
c
;
Zeid AlOthman
c
;
William A. Donald
d
;
Claudiu T. Supuran
c
;
d
;
e
;
claudiu.supuran@unifi.it
;
Clemente Capasso
a
;
clemente.capasso@ibbr.cnr.it
关键词:
Carbonic
anhydrase
;
γ-Class
;
Inhibitor
;
Sulfonamide
;
Sulfamate
;
Acetazolamide
;
Drug resistance
;
Burkholderia pseudomallei
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
3.
Dithiocarbamates effectively inhibit the β-
carbonic
anhydrase
from the dandruff-producing fungus Malassezia globosa
作者:
Daniela Vullo
a
;
Sonia Del Prete
b
;
c
;
Alessio Nocentini
b
;
Sameh M. Osman
d
;
Zeid AlOthman
d
;
Clemente Capasso
c
;
Murat Bozdag
a
;
Fabrizio Carta
b
;
Paola Gratteri
e
;
Claudiu T. Supuran
b
;
d
;
claudiu.supuran@unifi.it
关键词:
Carbonic
anhydrase
;
β-CA-class enzyme
;
Dithiocarbamate
;
Inhibitor
;
Malassezia globosa
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
4.
5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with effective
carbonic
anhydrase
inhibitor
y activity: Solution and crystallographic investigations
作者:
Jekaterīna Ivanova
a
;
b
;
Agnese Balode
a
;
b
;
Raivis Žalubovskis
a
;
raivis@osi.lv
;
Janis Leitans
c
;
Andris Kazaks
c
;
Daniela Vullo
d
;
Kaspars Tars
c
;
e
;
Claudiu T. Supuran
f
;
claudiu.supuran@unifi.it
关键词:
Carbonic
anhydrase
;
Thiophene-2-sulfonamide
;
Mercaptan
;
Inhibitor
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
5.
Novel eugenol derivatives: Potent acetylcholinesterase and
carbonic
anhydrase
inhibitor
s
作者:
Fevzi Topal
a
;
Ilhami Gulcin
b
;
c
;
igulcin@atauni.edu.tr
;
igulcin@yahoo.com
;
Arif Dastan
b
;
Murat Guney
d
关键词:
Eugenol
;
Carbonic
anhydrase
;
Acetylcholinesterase
;
Enzyme purification
;
Enzyme inhibition
刊名:International Journal of Biological Macromolecules
出版年:2017
6.
Substituted (E)-2-(2-benzylidenehydrazinyl)-4-methylthiazole-5-carboxylates as dual
inhibitor
s of 15-lipoxygenase &
carbonic
anhydrase
II: synthesis, biochemical evaluation and docking studies
作者:
Aamer Saeed
a
;
aamersaeed@yahoo.com
;
Shafi Ullah Khan
b
;
Parvez Ali Mahesar
a
;
Pervaiz Ali Channar
a
;
Ghulam Shabir
a
;
Jamshed Iqbal
b
;
drjamshed@ciit.net.pk
关键词:
Thiazoles
;
15-Lipoxygenase
;
Bovine
carbonic
anhydrase
II
;
Docking studies
刊名:Biochemical and Biophysical Research Communications
出版年:2017
7.
Anion inhibition profiles of the γ-
carbonic
anhydrase
from the pathogenic bacterium Burkholderia pseudomallei responsible of melioidosis and highly drug resistant to common antibiotics
作者:
Sonia Del Prete
a
;
b
;
Daniela Vullo
b
;
Pietro Di Fonzo
a
;
Sameh M. Osman
c
;
Zeid AlOthman
c
;
Claudiu T. Supuran
c
;
d
;
claudiu.supuran@unifi.it
;
Clemente Capasso
a
;
clemente.capasso@ibbr.cnr.it
关键词:
Carbonic
anhydrase
;
Metalloenzymes
;
γ-Class
;
Inhibitor
;
Anion
;
Burkholderia pseudomallei
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
8.
Carbonic
anhydrase
inhibition boosts the antitumor effects of Imatinib mesylate via potentiating the antiangiogenic and antimetastatic machineries
作者:
Amal A. Abd-El Fattah
a
;
Hebatallah A. Darwish
a
;
b
;
Nevine Fathy
a
;
nevine.abdallah@pharma.cu.edu.eg
;
Samia A. Shouman
c
关键词:
AZ
;
acetazolamide
;
IM
;
imatinib
;
EAC
;
Ehrlich ascites carcinoma
;
PDGF-A
;
platelet derived growth factor-A
;
TSP-1
;
thrombospondin-1
;
VEGF
;
vascular endothelial growth factor
;
NO
;
nitric oxide
;
MMP
;
matrix metalloproteinase
;
MAPK
;
mitogen activated protein kinase
;
TIMP
;
tissue
inhibitor
of metalloproteinase
;
MVD
;
microvessel density
刊名:Toxicology and Applied Pharmacology
出版年:2017
9.
New approach of delivering cytotoxic drugs towards CAIX expressing cells: A concept of dual-target drugs
作者:
Simon J.A. van Kuijk
a
;
1
;
s.vankuijk@maastrichtuniversity.nl
;
Nanda Kumar Parvathaneni
a
;
b
;
1
;
nanda-kumar.parvathaneni@etu.umontpellier.fr
;
Raymon Niemans
a
;
1
;
Marike W. van Gisbergen
a
;
1
;
Fabrizio Carta
c
;
Daniela Vullo
d
;
Silvia Pastorekova
e
;
Ala Yaromina
a
;
Claudiu T. Supuran
c
;
Ludwig J. Dubois
a
;
2
;
Jean-Yves Winum
b
;
2
;
Philippe Lambin
a
;
2
关键词:
Tumor
;
Hypoxia
;
Carbonic
anhydrase
IX
;
Dual-target drugs
;
CAIX
inhibitor
s
;
Cytotoxic drugs
刊名:European Journal of Medicinal Chemistry
出版年:2017
10.
Design and synthesis of a novel class of
carbonic
anhydrase
-IX
inhibitor
1-(3-(phenyl/4-fluorophenyl)-7-imino-3H-[1,2,3]triazolo[4,5d]pyrimidin 6(7H)yl)urea
作者:
Shikha Kumari
a
;
1
;
Danish Idrees
b
;
1
;
Chandra Bhushan Mishra
a
;
1
;
Amresh Prakash
b
;
1
;
Wahiduzzaman
b
;
Faizan Ahmad
b
;
Md. Imtaiyaz Hassan
b
;
mihassan@jmi.ac.in" class="auth_mail" title="E-mail the corresponding author
;
Manisha Tiwari
a
;
mtiwari07@gmail.com" class="auth_mail" title="E-mail the corresponding author
关键词:
Hypoxia-induced cancer
;
Carbonic
anhydrase
IX
inhibitor
;
Drug design and discovery
;
Triazolo-pyrimidine urea
;
MD simulation
刊名:Journal of Molecular Graphics and Modelling
出版年:2016
1
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4
5
6
7
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