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在“
ACS电子期刊
”中,
命中:
16
条,耗时:0.0609678 秒
在所有数据库中总计命中:
218
条
1.
Kin
a
se-Independent Sm
a
ll-Molecule Inhibition of JAK-STAT Sign
a
ling
作者:
D
a
nny Hung-Chieh Chou
;
A
medeo Vetere
;
A
mit Choudh
a
ry
;
Stephen S. Scully
;
Monic
a
Schenone
;
A
lici
a
T
a
ng
;
R
a
chel Gomez
;
Se
a
n M. Burns
;
Morten Lundh
;
T
a
m
a
r
a
Vit
a
l
;
E
a
mon Comer
;
P
a
trick W. F
a
loon
;
Vl
a
do D
a
n膷铆k
;
Christie Ci
a
rlo
;
Joshi
a
w
a
P
a
ulk
;
Mingji D
a
i
;
Cl
a
rk Reddy
;
H
a
nshi Sun
;
M
a
tthew Young
;
Nichol
a
s Don
a
to
;
J
a
cob J
a
ffe
;
P
a
ul A. Clemons
;
Michelle P
a
lmer
;
Steven
A
. C
a
rr
;
Stu
a
rt L. Schreiber
;
Bridget K. W
a
gner
刊名:Journ
a
l of the Americ
a
n Chemic
a
l Society
出版年:2015
2.
Combining X-r
a
y Cryst
a
llogr
a
phy
a
nd Molecul
a
r Modeling tow
a
rd the Optimiz
a
tion of Pyr
a
zolo[3,4-d]pyrimidines
a
s Potent c-Src Inhibitors Active in Vivo
a
g
a
inst Neurobl
a
stom
a
作者:
Cristin
a
Tintori
;
A
nn
a
Luci
a
F
a
ll
a
c
a
r
a
;
M
a
rco R
a
di
;
Cl
a
udio Z
a
mperini
;
Elen
a
Dre
a
ssi
;
Emm
a
nuele Cresp
a
n
;
Giov
a
nni M
a
g
a
;
Silvi
a
Schenone
;
Fr
a
ncesc
a
Musumeci
;
Chi
a
r
a
Brullo
;
A
ndr茅 Richters
;
Fr
a
ncesc
a
G
a
sp
a
rrini
;
A
dri
a
no Angelucci
;
Cl
a
udio Festucci
a
;
Simon
a
Delle Mon
a
che
;
D
a
niel R
a
uh
;
M
a
urizio Bott
a
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2015
3.
Studies on the
A
TP Binding Site of Fyn Kin
a
se for the Identific
a
tion of New Inhibitors
a
nd Their Ev
a
lu
a
tion
a
s Potenti
a
l Agents
a
g
a
inst T
a
uop
a
thies
a
nd Tumors
作者:
Cristin
a
Tintori
;
Giuseppin
a
L
a
S
a
l
a
;
Giuli
a
Vign
a
roli
;
Lorenzo Bott
a
;
A
nn
a
Luci
a
F
a
ll
a
c
a
r
a
;
Federico F
a
lchi
;
M
a
rco R
a
di
;
Cl
a
udio Z
a
mperini
;
Elen
a
Dre
a
ssi
;
Luci
a
Dello I
a
cono
;
Don
a
t
a
Orioli
;
Giuseppe Bi
a
monti
;
Mirko G
a
rbelli
;
A
ndre
a
Loss
a
ni
;
Fr
a
ncesc
a
G
a
sp
a
rrini
;
Tizi
a
no Tuccin
a
rdi
;
Il
a
ri
a
L
a
urenz
a
n
a
;
A
dri
a
no Angelucci
;
Giov
a
nni M
a
g
a
;
Silvi
a
Schenone
;
Chi
a
r
a
Brullo
;
Fr
a
ncesc
a
Musumeci
;
A
ndre
a
Desogus
;
Emm
a
nuele Cresp
a
n
;
M
a
urizio Bott
a
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2015
4.
Exploring the Chemic
a
l Sp
a
ce
a
round the Privileged Pyr
a
zolo[3,4-d]pyrimidine Sc
a
ffold: Tow
a
rd Novel Allosteric Inhibitors of T315I-Mut
a
ted Abl
作者:
Giuli
a
Vign
a
roli
;
M
a
rtin
a
Menc
a
relli
;
Debor
a
h Sement
a
;
Emm
a
nuele Cresp
a
n
;
Mirosl
a
v
a
Kissov
a
;
Giov
a
nni M
a
g
a
;
Silvi
a
Schenone
;
M
a
rco R
a
di
;
M
a
urizio Bott
a
刊名:
A
CS Combin
a
tori
a
l Science
出版年:2014
5.
Pyr
a
zolo[3,4-d]pyrimidine Prodrugs: Str
a
tegic Optimiz
a
tion of the Aqueous Solubility of Du
a
l Src/Abl Inhibitors
作者:
Giuli
a
Vign
a
roli
;
Cl
a
udio Z
a
mperini
;
Elen
a
Dre
a
ssi
;
M
a
rco R
a
di
;
A
dri
a
no Angelucci
;
P
a
trizi
a
S
a
nit脿
;
Emm
a
nuele Cresp
a
n
;
Mirosl
a
v
a
Kissov
a
;
Giov
a
nni M
a
g
a
;
Silvi
a
Schenone
;
Fr
a
ncesc
a
Musumeci
;
M
a
urizio Bott
a
刊名:
A
CS Medicin
a
l Chemistry Letters
出版年:2013
6.
In Silico Identific
a
tion
a
nd Biologic
a
l Ev
a
lu
a
tion of Novel Selective Serum/Glucocorticoid-Inducible Kin
a
se 1 Inhibitors B
a
sed on the Pyr
a
zolo-Pyrimidine Sc
a
ffold
作者:
Fr
a
ncesco Ortuso
;
Ros
a
rio Am
a
to
;
A
nn
a
Artese
;
Luci
a
D鈥檃nton
a
;
Giosu猫 Cost
a
;
Cristin
a
T
a
l
a
rico
;
Fr
a
ncesco Gigliotti
;
C
a
t
a
ldo Bi
a
nco
;
Fr
a
ncesco Tr
a
p
a
sso
;
Silvi
a
Schenone
;
Fr
a
ncesc
a
Musumeci
;
Lorenzo Bott
a
;
Nicol
a
Perrotti
;
Stef
a
no Alc
a
ro
刊名:Journ
a
l of Chemic
a
l Inform
a
tion
a
nd Modeling
出版年:2014
7.
Biologic
a
lly Driven Synthesis of Pyr
a
zolo[3,4-d]pyrimidines As Protein Kin
a
se Inhibitors: An Old Sc
a
ffold As
a
New Tool for Medicin
a
l Chemistry
a
nd Chemic
a
l Biology Studies
作者:
Silvi
a
Schenone
;
M
a
rco R
a
di
;
Fr
a
ncesc
a
Musumeci
;
Chi
a
r
a
Brullo
;
M
a
urizio Bott
a
刊名:Chemic
a
l Reviews
出版年:2014
8.
Insight into the
A
llosteric Inhibition of Abl Kin
a
se
作者:
A
nn
a
Luci
a
F
a
ll
a
c
a
r
a
;
Cristin
a
Tintori
;
M
a
rco R
a
di
;
Silvi
a
Schenone
;
M
a
urizio Bott
a
刊名:Journ
a
l of Chemic
a
l Inform
a
tion
a
nd Modeling
出版年:2014
9.
Design, Synthesis,
a
nd Biologic
a
l Ev
a
lu
a
tion of Pyr
a
zolo[3,4-d]pyrimidines Active in Vivo on the Bcr-Abl T315I Mut
a
nt
作者:
M
a
rco R
a
di
;
Cristin
a
Tintori
;
Fr
a
ncesc
a
Musumeci
;
Chi
a
r
a
Brullo
;
Cl
a
udio Z
a
mperini
;
Elen
a
Dre
a
ssi
;
A
nn
a
Luci
a
F
a
ll
a
c
a
r
a
;
Giuli
a
Vign
a
roli
;
Emm
a
nuele Cresp
a
n
;
S
a
m
a
nth
a
Z
a
noli
;
Il
a
ri
a
L
a
urenz
a
n
a
;
Irene Filippi
;
Giov
a
nni M
a
g
a
;
Silvi
a
Schenone
;
A
dri
a
no Angelucci
;
M
a
urizio Bott
a
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2013
10.
Identific
a
tion of New Fyn Kin
a
se Inhibitors Using
a
FLAP-B
a
sed Appro
a
ch
作者:
Giulio Poli
;
Tizi
a
no Tuccin
a
rdi
;
Fl
a
vio Rizzolio
;
Is
a
bell
a
C
a
ligiuri
;
Lorenzo Bott
a
;
C
a
rlott
a
Gr
a
nchi
;
G
a
briell
a
Ortore
;
Filippo Minutolo
;
Silvi
a
Schenone
;
A
dri
a
no M
a
rtinelli
刊名:Journ
a
l of Chemic
a
l Inform
a
tion
a
nd Modeling
出版年:2013
1
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