设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
Wiley电子期刊(13)
NATURE电子期刊(11)
ACS电子期刊(221)
SpringerLink电子期刊(320)
Elsevier电子期刊(1176)
在“
ACS电子期刊
”中,
命中:
221
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1,741
条
1.
Linear Free Energy Relationship Analysis of Transition State Mimicry by 3-Deoxy-d-arabino-heptulosonate-7-phosphate (DAHP) Oxime, a DAHP Synthase
Inhibitor
and Phosphate Mimic
作者:
Naresh Balachandran
;
Frederick ToPaul J. Berti
刊名:Biochemistry
出版年:2017
2.
Covalent Guanosine Mimetic
Inhibitor
s of G12C KRAS
作者:
Yuan Xiong
;
Jia Lu
;
John Hunter
;
Lianbo Li
;
David Scott
;
Hwan Geun Choi
;
Sang Min Lim
;
Anuj Manandhar
;
Sudershan Gondi
;
Taebo Sim
;
Kenneth D. Westover
;
Nathanael S. Gray
刊名:ACS Medicinal Chemistry Letters
出版年:2017
3.
The Structure of Murine N1-Acetylspermine Oxidase Reveals Molecular Details of Vertebrate Polyamine Catabolism
作者:
Tove SjögrenCarola M. Wassvik
;
Arjan Snijder
;
Anna Aagaard
;
Taichi Kumanomidou
;
Louise Barlind
;
Tim P. Kaminski
;
Akiko Kashima
;
Takehiro Yokota
;
Ola Fjellström
刊名:Biochemistry
出版年:2017
4.
Triazole Ureas Act as Diacylglycerol Lipase
Inhibitor
s and Prevent Fasting-Induced Refeeding
作者:
Hui DengSander Kooijman
;
Adrianus M. C. H. van den Nieuwendijk
;
Daisuke Ogasawara
;
Tom van der Wel
;
Floris van Dalen
;
Marc P. Baggelaar
;
Freek J. JanssenRichard J. B. H. N. van den Berg
;
Hans den Dulk
;
Benjamin F. Cravatt
;
Herman S. Overkleeft
;
Patrick C. N. RensenMario van der Stelt
刊名:Journal of Medicinal Chemistry
出版年:2017
5.
Discovery of 1-{(3R,4R)-3-[({5-Chloro-2-[(1-methyl-1H-pyrazol-4-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Potent, WT Sparing,
Irreversible
Inhibitor
of T790M-Containing EGFR Mutants
作者:
Hengmiao Cheng
;
Sajiv K. Nair
;
Brion W. Murray
;
Chau Almaden
;
Simon Bailey
;
Sangita Baxi
;
Doug Behenna
;
Sujin Cho-Schultz
;
Deepak Dalvie
;
Dac M. Dinh
;
Martin P. Edwards
;
Jun Li Feng
;
Rose Ann Ferre
;
Ketan S. Gajiwala
;
Michelle D. Hemkens
;
Amy Jackson-Fisher
;
Mehran Jalaie
;
Ted O. Johnson
;
Robert S. Kania
;
Susan Kephart
;
Jennifer Lafontaine
;
Beth Lunney
;
Kevin K.-C. Liu
;
Zhengyu Liu
;
Jean Matthews
;
Asako Nagata
;
Sherry Niessen
;
Martha A. Ornelas
;
Suvi T. M. Orr
;
Mason Pairish
;
Simon Planken
;
Shijian Ren
;
Daniel Richter
;
Kevin Ryan
;
Neal Sach
;
Hong Shen
;
Tod Smeal
;
Jim Solowiej
;
Scott Sutton
;
Khanh Tran
;
Elaine Tseng
;
William Vernier
;
Marlena Walls
;
Shuiwang Wang
;
Scott L. Weinrich
;
Shuibo Xin
;
Haiwei Xu
;
Min-Jean Yin
;
Michael Zientek
;
Ru Zhou
;
John C. Kath
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Spiroepoxytriazoles Are Fumagillin-like
Irreversible
Inhibitor
s of MetAP2 with Potent Cellular Activity
作者:
Michael Morgen
;
Christian Jöst
;
Mona Malz
;
Robert Janowski
;
Dierk Niessing
;
Christian D. Klein
;
Nikolas Gunkel
;
Aubry K. Miller
刊名:ACS Chemical Biology
出版年:2016
7.
Development of Specific,
Irreversible
Inhibitor
s for a Receptor Tyrosine Kinase EphB3
作者:
Alvin Kung
;
Ying-Chu Chen
;
Marianne Schimpl
;
Feng Ni
;
Jianfa Zhu
;
Maurice Turner
;
Henrik Molina
;
Ross Overman
;
Chao Zhang
刊名:Journal of the American Chemical Society
出版年:2016
8.
Structure–Activity Relationship of 18F-Labeled Phosphoramidate Peptidomimetic Prostate-Specific Membrane Antigen (PSMA)-Targeted
Inhibitor
Analogues for PET Imaging of Prostate Cancer
作者:
Shorouk Dannoon
;
Tanushree Ganguly
;
Hendry Cahaya
;
Jonathan J. Geruntho
;
Matthew S. Galliher
;
Sophia K. Beyer
;
Cindy J. Choy
;
Mark R. Hopkins
;
Melanie Regan
;
Joseph E. Blecha
;
Lubica Skultetyova
;
Christopher R. Drake
;
Salma Jivan
;
Cyril Barinka
;
Ella F. Jones
;
Clifford E. Berkman
;
Henry F. VanBrocklin
刊名:Journal of Medicinal Chemistry
出版年:2016
9.
Synthesis and Preliminary PET Imaging Studies of a FAAH Radiotracer ([11C]MPPO) Based on α-Ketoheterocyclic Scaffold
作者:
Lu Wang
;
Joji Yui
;
Qifan Wang
;
Yiding Zhang
;
Wakana Mori
;
Yoko Shimoda
;
Masayuki Fujinaga
;
Katsushi Kumata
;
Tomoteru Yamasaki
;
Akiko Hatori
;
Benjamin H. Rotstein
;
Thomas Lee Collier
;
Chongzhao Ran
;
Neil Vasdev
;
Ming-Rong Zhang
;
Steven H. Liang
刊名:ACS Chemical Neuroscience
出版年:2016
10.
Identification of SNAIL1 Peptide-Based
Irreversible
Lysine-Specific Demethylase 1-Selective Inactivators
作者:
Yukihiro Itoh
;
Keisuke Aihara
;
Paolo Mellini
;
Toshifumi Tojo
;
Yosuke Ota
;
Hiroki Tsumoto
;
Viswas Raja Solomon
;
Peng Zhan
;
Miki Suzuki
;
Daisuke Ogasawara
;
Akira Shigenaga
;
Tsubasa Inokuma
;
Hidehiko Nakagawa
;
Naoki Miyata
;
Tamio Mizukami
;
Akira Otaka
;
Takayoshi Suzuki
刊名:Journal of Medicinal Chemistry
出版年:2016
1
2
3
4
5
6
7
8
9
按检索点细分(221)
刊名(18)
作者(3)
关键词(194)
按出版年细分(221)
2017年(4)
2016年(14)
2015年(8)
2014年(17)
2013年(22)
2012年(17)
2011年(7)
2010年(4)
2009年(10)
2008年(10)
2007年(11)
2006年(9)
2005年(12)
2004年(5)
2003年(9)
2002年(3)
2001年(13)
2000年(7)
2000年及以前(39)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.