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NATURE电子期刊(1)
Elsevier电子期刊(10)
ACS电子期刊(14)
在“
ACS电子期刊
”中,
命中:
14
条,耗时:小于0.01 秒
在所有数据库中总计命中:
25
条
1.
Characterizing the Epothilone Binding Site on β-Tubulin by Photoaffinity Labeling: Identification of β-Tubulin Peptides TARGSQQY and TSRGSQQY as Targets of an Epothilone Photoprobe for Polymerized Tubulin
作者:
Adwait R. Ranade
;
LeeAnn Higgins
;
Todd W. Markowski
;
Nicole Glaser
;
Dmitry Kashin
;
Ruoli
Bai
;
Kwon Ho Hong
;
Ernest Hamel
;
Gerhard Höfle
;
Gunda I. Georg
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Novel Microtubule-Targeting 7-Deazahypoxanthines Derived from Marine Alkaloid Rigidins with Potent in Vitro and in Vivo Anticancer Activities
作者:
Derek C. Medellin
;
Qiong Zhou
;
Robert Scott
;
R. Matthew Hill
;
Sarah K. Frail
;
Ramesh Dasari
;
Steven J. Ontiveros
;
Stephen C. Pelly
;
Willem A. L. van Otterlo
;
Tania Betancourt
;
Charles B. Shuster
;
Ernest Hamel
;
Ruoli
Bai
;
Daniel V. LaBarbera
;
Snezna Rogelj
;
Liliya V. Frolova
;
Alexander Kornienko
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Dependent Cancer
作者:
Giuseppe La Regina
;
Ruoli
Bai
;
Antonio Coluccia
;
Valeria Famiglini
;
Sveva Pelliccia
;
Sara Passacantilli
;
Carmela Mazzoccoli
;
Vitalba Ruggieri
;
Annalisa Verrico
;
Andrea Miele
;
Ludovica Monti
;
Marianna Nalli
;
Romina Alfonsi
;
Lucia Di Marcotullio
;
Alberto Gulino
;
Biancamaria Ricci
;
Alessandra Soriani
;
Angela Santoni
;
Michele Caraglia
;
Stefania Porto
;
Eleonora Da Pozzo
;
Claudia Martini
;
Andrea Brancale
;
Luciana Marinelli
;
Ettore Novellino
;
Stefania Vultaggio
;
Mario Varasi
;
Ciro Mercurio
;
Chiara Bigogno
;
Giulio Dondio
;
Ernest Hamel
;
Patrizia Lavia
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Discovery of Biarylaminoquinazolines as Novel Tubulin Polymerization Inhibitors
作者:
Giovanni Marzaro
;
Antonio Coluccia
;
Alessandro Ferrarese
;
Paola Brun
;
Ignazio Castagliuolo
;
Maria Teresa Conconi
;
Giuseppe La Regina
;
Ruoli
Bai
;
Romano Silvestri
;
Ernest Hamel
;
Adriana Chilin
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
New Pyrrole Derivatives with Potent Tubulin Polymerization Inhibiting Activity As Anticancer Agents Including Hedgehog-Dependent Cancer
作者:
Giuseppe La Regina
;
Ruoli
Bai
;
Antonio Coluccia
;
Valeria Famiglini
;
Sveva Pelliccia
;
Sara Passacantilli
;
Carmela Mazzoccoli
;
Vitalba Ruggieri
;
Lorenza Sisinni
;
Alessio Bolognesi
;
Whilelmina Maria Rensen
;
Andrea Miele
;
Marianna Nalli
;
Romina Alfonsi
;
Lucia Di Marcotullio
;
Alberto Gulino
;
Andrea Brancale
;
Ettore Novellino
;
Giulio Dondio
;
Stefania Vultaggio
;
Mario Varasi
;
Ciro Mercurio
;
Ernest Hamel
;
Patrizia Lavia
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
Toward Highly Potent Cancer Agents by Modulating the C-2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors
作者:
Giuseppe La Regina
;
Ruoli
Bai
;
Whilelmina Maria Rensen
;
Erica Di Cesare
;
Antonio Coluccia
;
Francesco Piscitelli
;
Valeria Famiglini
;
Alessia Reggio
;
Marianna Nalli
;
Sveva Pelliccia
;
Eleonora Da Pozzo
;
Barbara Costa
;
Ilaria Granata
;
Amalia Porta
;
Bruno Maresca
;
Alessandra Soriani
;
Maria Luisa Iannitto
;
Angela Santoni
;
Junjie Li
;
Marlein Miranda Cona
;
Feng Chen
;
Yicheng Ni
;
Andrea Brancale
;
Giulio Dondio
;
Stefania Vultaggio
;
Mario Varasi
;
Ciro Mercurio
;
Claudia Martini
;
Ernest Hamel
;
Patrizia Lavia
;
Ettore Novellino
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Steroidomimetic Tetrahydroisoquinolines for the Design of New Microtubule Disruptors
作者:
Mathew P. Leese
;
Fabrice Jourdan
;
Wolfgang Dohle
;
Meriel R. Kimberley
;
Mark P. Thomas
;
Ruoli
Bai
;
Ernest Hamel
;
Eric Ferrandis
;
Barry V. L. Potter
刊名:ACS Medicinal Chemistry Letters
出版年:2012
8.
Design and Synthesis of 2-Heterocyclyl-3-arylthio-1H-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability
作者:
Giuseppe La Regina
;
Ruoli
Bai
;
Willeke Rensen
;
Antonio Coluccia
;
Francesco Piscitelli
;
Valerio Gatti
;
Alessio Bolognesi
;
Antonio Lavecchia
;
Ilaria Granata
;
Amalia Porta
;
Bruno Maresca
;
Alessandra Soriani
;
Maria Luisa Iannitto
;
Marisa Mariani
;
Angela Santoni
;
Andrea Brancale
;
Cristiano Ferlini
;
Giulio Dondio
;
Mario Varasi
;
Ciro Mercurio
;
Ernest Hamel
;
Patrizia Lavia
;
Ettore Novellino
;
Romano Silvestri
刊名:Journal of Medicinal Chemistry
出版年:2011
9.
Interactions of Halichondrin B and Eribulin with Tubulin
作者:
Ruoli
Bai
;
Tam Luong Nguyen
;
James C. Burnett
;
Onur Atasoylu
;
Murray H. G. Munro
;
George R. Pettit
;
Amos B. Smith
;
III
;
Rick Gussio
;
Ernest Hamel
刊名:Journal of Chemical Information and Modeling
出版年:2011
10.
New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies
作者:
Giuseppe La Regina
;
Taradas Sarkar
;
Ruoli
Bai
;
Michael C. Edler
;
Roberto Saletti
;
Antonio Coluccia
;
Francesco Piscitelli
;
Lara Minelli
;
Valerio Gatti
;
Carmela Mazzoccoli
;
Vanessa Palermo
;
Cristina Maz
刊名:Journal of Medicinal Chemistry
出版年:2009
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