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SpringerLink电子期刊(5)
Elsevier电子期刊(76)
ACS电子期刊(12)
在“
ACS电子期刊
”中,
命中:
12
条,耗时:0.0479808 秒
在所有数据库中总计命中:
93
条
1.
Iden
t
ifica
t
ion and Preclinical Pharmacolo
g
y of BMS-986104: A Differen
t
ia
t
ed S1P1 Recep
t
or Modula
t
or in Clinical Trials
作者:
T
.
G
.
Murali
Dhar
;
Hai-Yun Xiao
;
Jenny Xie
;
Lois D. Lehman-McKeeman
;
Dauh-Rurn
g
Wu
;
Mar
t
a Dabros
;
Xiaoxia Yan
g
;
T
racy L. Taylor
;
Xia D. Zhou
;
Elizabe
t
h M. Heimrich
;
Rochelle
T
homas
;
Kim W. McIn
t
yre
;
Be
t
hanne Warrack
;
Hon
g
Shi
;
Paul C. Levesque
;
Jia L. Zhu
;
James Hennan
;
Praveen Balimane
;
Zhen
g
Yan
g
;
An
t
hony M. Marino
;
G
eor
g
ia Cornelius
;
Celia J. D’Arienzo
;
Arvind Ma
t
hur
;
Din
g
Ren Shen
;
Mary Ellen Cvijic
;
Luisa Sal
t
er-Cid
;
Joel C. Barrish
;
Percy H. Car
t
er
;
Alaric J. Dyckman
刊名:ACS Medicinal Chemis
t
ry Le
tt
ers
出版年:2016
2.
Asymme
t
ric Hydrobora
t
ion Approach
t
o
t
he Scalable Syn
t
hesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-
t
e
t
rahydronaph
t
halen-2-yl)cyclopen
t
yl)me
t
hanol (BMS-986104) as a Po
t
en
t
S1P1 Recep
t
or Modula
t
or
作者:
Michael
G
. Yan
g
Zili Xiao
;
T
.
G
.
Murali
Dhar
;
Hai-Yun Xiao
;
John L.
G
ilmore
;
David Marcoux
;
Jenny H. Xie
;
Kim W. McIn
t
yre
;
T
racy L. Taylor
;
Virna Borowski
;
Elizabe
t
h Heimrich
;
Yu-Wen Li
;
Jianlin Fen
g
;
Alda Fernandes
;
Zhen
g
Yan
g
;
Praveen Balimane
;
An
t
hony M. Marino
;
G
eor
g
ia Cornelius
;
Be
t
hanne M. Warrack
;
Arvind Ma
t
hur
;
Dauh-Rurn
g
Wu
;
Pen
g
Li
;
Anuradha
G
up
t
a
;
Bala Pra
g
ala
t
han
;
Din
g
Ren Shen
;
Mary Ellen Cvijic
;
Lois D. Lehman-McKeeman
;
Luisa Sal
t
er-Cid
;
Joel C. Barrish
;
Percy H. Car
t
er
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemis
t
ry
出版年:2016
3.
Discovery of ((4-(5-(Cyclopropylcarbamoyl)-2-me
t
hylphenylamino)-5-me
t
hylpyrrolo[1,2-f][1,2,4]
t
riazine-6-carbonyl)(propyl)carbamoyloxy)me
t
hyl-2-(4-(phosphonooxy)phenyl)ace
t
a
t
e聽(BMS-751324), a Cl
作者:
Chunjian Liu
;
James Lin
;
John Hynes
;
Hon
g
Wu
;
S
t
ephen T. Wrobleski
;
Shuqun Lin
;
T
.
G
.
Murali
Dhar
;
Vivekananda M. Vrudhula
;
Jun
g
-Hui Sun
;
Sam Chao
;
Rulin Zhao
;
Bei Wan
g
;
Ban
g
-Chi Chen
;
G
erry Everlof
;
Chris
t
oph
G
esenber
g
;
Hon
g
jian Zhan
g
;
Puni
t
H. Mara
t
he
;
Kim W. McIn
t
yre
;
T
racy L. Taylor
;
Ka
t
hleen
G
illooly
;
David J. Shus
t
er
;
Murray McKinnon
;
John H. Dodd
;
Joel C. Barrish
;
G
ary L. Schieven
;
Ka
t
erina Lef
t
heris
刊名:Journal of Medicinal Chemis
t
ry
出版年:2015
4.
Iden
t
ifica
t
ion of Tricyclic A
g
onis
t
s of Sphin
g
osine-1-phospha
t
e Recep
t
or 1 (S1P1) Employin
g
Li
g
and-Based Dru
g
Desi
g
n
作者:
Hai-Yun Xiao
;
Sco
tt
H. Wa
tt
erson
;
Charles M. Lan
g
evine
;
Anura
g
S. Srivas
t
ava
;
Soo S. Ko
;
Yanlei Zhan
g
;
Rober
t
J. Cherney
;
Wei-Wei
G
uo
;
John L.
G
ilmore
;
James E. Sheppeck II
;
Dauh-Rurn
g
Wu
;
Pen
g
Li
;
Duraisamy Ramasamy
;
Piramanaya
g
am Arunachalam
;
Arvind Ma
t
hur
;
T
racy L. Taylor
;
David J. Shus
t
er
;
Kim W. McIn
t
yre
;
Din
g
-Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
An
t
hony M. Marino
;
Praveen V. Balimane
;
Zhen
g
Yan
g
;
Dana M. Banas
;
G
eor
g
ia Cornelius
;
Celia J. D’Arienzo
;
Be
t
hanne M. Warrack
;
Lois Lehman-McKeeman
;
Luisa M. Sal
t
er-Cid
;
Jenny Xie
;
Joel C. Barrish
;
Percy H. Car
t
er
;
Alaric J. Dyckman
;
T
.
G
.
Murali
Dhar
刊名:Journal of Medicinal Chemis
t
ry
出版年:2016
5.
Improvin
g
t
he Pharmacokine
t
ic and CYP Inhibi
t
ion Profiles of Azaxan
t
hene-Based Glucocor
t
icoid Recep
t
or Modula
t
ors鈥擨den
t
ifica
t
ion of (S)-5-(2-(9-Fluoro-2-(4-(2-hydroxypropan-2-yl)phenyl)-5H
作者:
Michael
G
. Yan
g
;
T
.
G
.
Murali
Dhar
;
Zili Xiao
;
Hai-Yun Xiao
;
James J.-W. Duan
;
Bin Jian
g
;
Michael A.
G
alella
;
Mark Cunnin
g
ham
;
Jinhon
g
Wan
g
;
Sium Hab
t
e
;
David Shus
t
er
;
Kim W. McIn
t
yre
;
Julie Carman
;
Deborah A. Holloway
;
John E. Somerville
;
S
t
even
G
. Nadler
;
Luisa Sal
t
er-Cid
;
Joel C. Barrish
;
David S. Weins
t
ein
刊名:Journal of Medicinal Chemis
t
ry
出版年:2015
6.
A New and Efficien
t
Syn
t
hesis of 6-[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-me
t
hyl-2,4-dioxo-1,3,7-
t
riazaspiro[4.4]non-7-yl]nico
t
inic Acid, a Po
t
en
t
LFA-1/ICAM Inhibi
t
or
作者:
Huipin
g
Zhan
g
;
Sco
tt
H. Wa
tt
erson
;
Zili Xiao
;
T
.
G
.
Murali
Dhar
;
Balu Balasubramanian
;
Joel C. Barrish
;
Ban
g
-Chi Chen
刊名:Or
g
anic Process Research & Developmen
t
出版年:2010
7.
Novel Syn
t
hesis of
t
he Hexahydroimidazo[1,5b]isoquinoline Scaffold: Applica
t
ion
t
o
t
he Syn
t
hesis of
G
lucocor
t
icoid Recep
t
or Modula
t
ors
作者:
Hai-Yun Xiao
;
Dauh-Rurn
g
Wu
;
Mary F. Malley
;
Jack Z.
G
ou
g
ou
t
as
;
Sium F. Hab
t
e
;
Mark D. Cunnin
g
ham
;
John E. Somerville
;
John H. Dodd
;
Joel C. Barrish
;
S
t
even
G
. Nadler
;
T
.
G
.
Murali
Dhar
刊名:Journal of Medicinal Chemis
t
ry
出版年:2010
8.
Acridone-Based Inhibi
t
ors of Inosine 5'-Monophospha
t
e Dehydro
g
enase: Discovery and SAR Leadin
g
t
o
t
he Iden
t
ifica
t
ion of N-(2-(6-(4-E
t
hylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2- fluoro-9-oxo-
作者:
Sco
tt
H. Wa
tt
erson
;
Pin
g
Chen
;
Yufen Zhao
;
Henry H.
G
u
;
T
.
G
.
Murali
Dhar
;
Zili Xiao
;
Shelley K. Ballen
t
ine
;
Zhon
g
qi Shen
;
Ca
t
herine A. Fleener
;
Ka
t
herine A. Rouleau
;
Mary Obermeier
;
Zhen
g
Yan
g
;
Kim W
刊名:Journal of Medicinal Chemis
t
ry
出版年:2007
9.
Ca
t
aly
t
ic Func
t
ionali
t
ies of H--Zeoli
t
e-Suppor
t
ed Molybdenum Hydro
t
rea
t
in
g
Ca
t
alys
t
s
作者:
G
. Mu
t
hu Kumaran
;
Shelu
G
ar
g
;
Kapil Soni
;
V. V. D. N. Prasad
;
L. D. Sharma
;
G
.
Murali
Dhar
刊名:Ener
g
y & Fuels
出版年:2006
10.
Effec
t
of Al-SBA-15 Suppor
t
on Ca
t
aly
t
ic Func
t
ionali
t
ies of Hydro
t
rea
t
in
g
Ca
t
alys
t
s. II. Effec
t
of Varia
t
ion of Molybdenum and Promo
t
er Con
t
en
t
s on Ca
t
aly
t
ic Func
t
ionali
t
ies
作者:
G
. Mu
t
hu Kumaran
;
Shelu
G
ar
g
;
Kapil Soni
;
Manoj Kumar
;
L. D. Sharma
;
K. S. Rama Rao
;
G
.
Murali
Dhar
刊名:Indus
t
rial & En
g
ineerin
g
Chemis
t
ry Research
出版年:2007
1
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