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1.
8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors
作者:
Vassilios Bavetsias
;
Rachel M. Lanigan
;
Gian Filippo Ruda
;
Butrus Atrash
;
Mark G. McLaughlin
;
Anthony Tumber
;
N. Yi Mok
;
Yann-Vaï Le Bihan
;
Sally Dempster
;
Katherine J. Boxall
;
Fiona Jeganathan
;
Stephanie B. Hatch
;
Pavel Savitsky
;
Srikannathasan Velupillai
;
Tobias Krojer
;
Katherine S. England
;
Jimmy Sejberg
;
Ching Thai
;
Adam
Donovan
;
Akos Pal
;
Giuseppe Scozzafava
;
James M. Bennett
;
Akane Kawamura
;
Catrine Johansson
;
Aleksandra Szykowska
;
Carina Gileadi
;
Nicola A. Burgess-Brown
;
Frank von Delft
;
Udo Oppermann
;
Zoe Walters
;
Janet Shipley
;
Florence I. Raynaud
;
Susan M. Westaway
;
Rab K. Prinjha
;
Oleg Fedorov
;
Rosemary Burke
;
Christopher J. Schofield
;
Isaac M. Westwood
;
Chas Bountra
;
Susanne Müller
;
Rob L. M. van Montfort
;
Paul E. Brennan
;
Julian Blagg
刊名:Journal of Medicinal Chemistry
出版年:2016
1
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