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知网期刊论文(1)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1
条
1.
Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials
作者:
T. G. Murali Dhar
;
Hai-Yun Xiao
;
Jenny Xie
;
Lois D. Lehman-McKeeman
;
Dauh-Rurng Wu
;
Marta Dabros
;
Xiaoxia Yang
;
Tracy L. Taylor
;
Xia D. Zhou
;
Elizabeth M. Heimrich
;
Rochelle Thomas
;
Kim W. McIntyre
;
Bethanne Warrack
;
Hong Shi
;
Paul C. Levesque
;
Jia L. Zhu
;
James Hennan
;
Praveen Balimane
;
Zheng Yang
;
Anthony M. Marino
;
Georgia Cornelius
;
Celia J. D’Arienzo
;
Arvind Mathur
;
Ding Ren Shen
;
Mary
Ellen
Cvijic
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery and Structure–Activity Relationship (SAR) of a Series of Ethanolamine-Based Direct-Acting Agonists of Sphingosine-1-phosphate (S1P1)
作者:
John L. Gilmore
;
James E. Sheppeck II
;
Scott H. Watterson
;
Lauren Haque
;
Parag Mukhopadhyay
;
Andrew J. Tebben
;
Michael A. Galella
;
Ding Ren Shen
;
Melissa Yarde
;
Mary
Ellen
Cvijic
;
Virna Borowski
;
Kathleen Gillooly
;
Tracy Taylor
;
Kim W. McIntyre
;
Bethanne Warrack
;
Paul C. Levesque
;
Julia P. Li
;
Georgia Cornelius
;
Celia D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Luisa Salter-Cid
;
Joel C. Barrish
;
William J. Pitts
;
Percy H. Carter
;
Jenny Xie
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Potent and Selective Agonists of Sphingosine 1-Phosphate 1 (S1P1): Discovery and SAR of a Novel Isoxazole Based Series
作者:
Scott H. Watterson
;
Junqing Guo
;
Steve H. Spergel
;
Charles M. Langevine
;
Robert V. Moquin
;
Ding Ren Shen
;
Melissa Yarde
;
Mary
Ellen
Cvijic
;
Dana Banas
;
Richard Liu
;
Suzanne J. Suchard
;
Kathleen Gillooly
;
Tracy Taylor
;
Sandra Rex-Rabe
;
David J. Shuster
;
Kim W. McIntyre
;
Georgia Cornelius
;
Celia D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Bethanne Warrack
;
Luisa Salter-Cid
;
Murray McKinnon
;
Joel C. Barrish
;
Percy H. Carter
;
William J. Pitts
;
Jenny Xie
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P1 Receptor Modulator
作者:
Michael G. YangZili Xiao
;
T. G. Murali Dhar
;
Hai-Yun Xiao
;
John L. Gilmore
;
David Marcoux
;
Jenny H. Xie
;
Kim W. McIntyre
;
Tracy L. Taylor
;
Virna Borowski
;
Elizabeth Heimrich
;
Yu-Wen Li
;
Jianlin Feng
;
Alda Fernandes
;
Zheng Yang
;
Praveen Balimane
;
Anthony M. Marino
;
Georgia Cornelius
;
Bethanne M. Warrack
;
Arvind Mathur
;
Dauh-Rurng Wu
;
Peng Li
;
Anuradha Gupta
;
Bala Pragalathan
;
Ding Ren Shen
;
Mary
Ellen
Cvijic
;
Lois D. Lehman-McKeeman
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug Design
作者:
Hai-Yun Xiao
;
Scott H. Watterson
;
Charles M. Langevine
;
Anurag S. Srivastava
;
Soo S. Ko
;
Yanlei Zhang
;
Robert J. Cherney
;
Wei-Wei Guo
;
John L. Gilmore
;
James E. Sheppeck II
;
Dauh-Rurng Wu
;
Peng Li
;
Duraisamy Ramasamy
;
Piramanayagam Arunachalam
;
Arvind Mathur
;
Tracy L. Taylor
;
David J. Shuster
;
Kim W. McIntyre
;
Ding-Ren Shen
;
Melissa Yarde
;
Mary
Ellen
Cvijic
;
Anthony M. Marino
;
Praveen V. Balimane
;
Zheng Yang
;
Dana M. Banas
;
Georgia Cornelius
;
Celia J. D’Arienzo
;
Bethanne M. Warrack
;
Lois Lehman-McKeeman
;
Luisa M. Salter-Cid
;
Jenny Xie
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
;
T. G. Murali Dhar
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors
作者:
Ashvinikumar V. Gavai
;
Claude Quesnelle
;
Derek Norris
;
Wen-Ching Han
;
Patrice Gill
;
Weifang Shan
;
Aaron Balog
;
Ke Chen
;
Andrew Tebben
;
Richard Rampulla
;
Dauh-Rurng Wu
;
Yingru Zhang
;
Arvind Mathur
;
Ronald White
;
Anne Rose
;
Haiqing Wang
;
Zheng Yang
;
Asoka Ranasinghe
;
Celia D鈥橝rienzo
;
Victor Guarino
;
Lan Xiao
;
Ching Su
;
Gerry Everlof
;
Vinod Arora
;
Ding Ren Shen
;
Mary
Ellen
Cvijic
;
Krista Menard
;
Mei-Li Wen
;
Jere Meredith
;
George Trainor
;
Louis J. Lombardo
;
Richard Olson
;
Phil S. Baran
;
John T. Hunt
;
Gregory D. Vite
;
Bruce S. Fischer
;
Richard A. Westhouse
;
Francis Y. Lee
刊名:ACS Medicinal Chemistry Letters
出版年:2015
7.
Discovery of a Potent and Orally Bioavailable Dual Antagonist of CC Chemokine Receptors 2 and 5
作者:
Percy H. Carter
;
Gregory D. Brown
;
Robert J. Cherney
;
Douglas G. Batt
;
Jing Chen
;
Cheryl M. Clark
;
Mary
Ellen
Cvijic
;
John V. Duncia
;
Soo S. Ko
;
Sandhya Mandlekar
;
Ruowei Mo
;
David J. Nelson
;
Jian Pang
;
Anne V. Rose
;
Joseph B. Santella
;
III
;
Andrew J. Tebben
;
Sarah C. Traeger
;
Songmei Xu
;
Qihong Zhao
;
Joel C. Barrish
刊名:ACS Medicinal Chemistry Letters
出版年:2015
8.
Discovery of the CCR1 Antagonist, BMS-817399, for the Treatment of Rheumatoid Arthritis
作者:
Joseph B. Santella
;
III
;
Daniel S. Gardner
;
John V. Duncia
;
Hong Wu
;
Murali Dhar
;
Cullen Cavallaro
;
Andrew J. Tebben
;
Percy H. Carter
;
Joel C. Barrish
;
Melissa Yarde
;
Stephanie W. Briceno
;
Mary
Ellen
Cvijic
;
R. Robert Grafstrom
;
Richard Liu
;
Sima R. Patel
;
Andrew J. Watson
;
Guchen Yang
;
Anne V. Rose
;
Rodney D. Vickery
;
Janet Caceres-Cortes
;
Christian Caporuscio
;
Daniel M. Camac
;
Javed A. Khan
;
Yongmi An
;
William R. Foster
;
Paul Davies
;
John Hynes
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
9.
Solid Phase Synthesis of 1,5-Diarylpyrazole-4-carboxamides: Discovery of Antagonists of the CB-1 Receptor
作者:
Annapurna Pendri
;
Dharmpal S. Dodd
;
Jing Chen
;
Mary
Ellen
Cvijic
;
Liya Kang
;
Rose A. Baska
;
Kenneth E. Carlson
;
Neil T. Burford
;
Chongqing Sun
;
William R. Ewing
;
Samuel W. Gerritz
刊名:ACS Combinatorial Science
出版年:2012
10.
Discovery and Lead Optimization of a Novel Series of CC Chemokine Receptor 1 (CCR1)-Selective Piperidine Antagonists via Parallel Synthesis
作者:
Cullen L. Cavallaro
;
Stephanie Briceno
;
Jing Chen
;
Mary
Ellen
Cvijic
;
Paul Davies
;
John Hynes
;
Jr.
;
Rui-Qin Liu
;
Sandhya Mandlekar
;
Anne V. Rose
;
Andrew J. Tebben
;
Katy Van Kirk
;
Andrew Watson
;
Hong Wu
;
Guchen Yang
;
Percy H. Carter
刊名:Journal of Medicinal Chemistry
出版年:2012
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