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ACS电子期刊(69)
在“
ACS电子期刊
”中,
命中:
69
条,耗时:0.0459441 秒
在所有数据库中总计命中:
4,184
条
1.
Discovery of (S)-
1
-(
1
-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((
1
-methyl-
1
H-pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(
1
H)-one (GDC-0994), an Extracellular Signal-Regulated
Kinase
1
/2 (ERK
1
/2) Inhibitor in Early Clinical Development
作者:
James F. Blake
;
Michael Burkard
;
Jocelyn Chan
;
Huifen Chen
;
Kang-Jye Chou
;
Dolores Diaz
;
Danette A. Dudley
;
John J. Gaudino
;
Stephen E. Gould
;
Jonas Grina
;
Thomas Hunsaker
;
Lichuan Liu
;
Matthew Martinson
;
David Moreno
;
Lars Mueller
;
Christine Orr
;
Patricia Pacheco
;
Ann Qin
;
Kevin Rasor
;
Li Ren
;
Kirk Robarge
;
Sheerin Shahidi-Latham
;
Jeffrey Stults
;
Francis Sullivan
;
Weiru Wang
;
Jianping Yin
;
Aihe Zhou
;
Marcia Belvin
;
Mark Merchant
;
John Moffat
;
Jacob B. Schwarz
刊名:Journal of Medicinal Chemistry
出版年:20
1
6
2.
Discovery of Bifunctional Oncogenic Target Inhibitors against Allosteric Mitogen-Activated Protein
Kinase
(
MEK1
) and Phosphatidylinositol 3-Kinase (PI3K)
作者:
Marcian E. Van Dort
;
Hao Hong
;
Hanxiao Wang
;
Charles A. Nino
;
Rachel L. Lombardi
;
Avery E. Blanks
;
Stefanie Galbán
;
Brian D. Ross
刊名:Journal of Medicinal Chemistry
出版年:20
1
6
3.
Discovery of
1
-(
1
H-Pyrazolo[4,3-c]pyridin-6-yl)urea Inhibitors of Extracellular Signal-Regulated
Kinase
(ERK) for the Treatment of Cancers
作者:
Jongwon Lim
;
Elizabeth H. Kelley
;
Joey L. Methot
;
Hua Zhou
;
Alessia Petrocchi
;
Hongmin Chen
;
Susan E. Hill
;
Marlene C. Hinton
;
Alan Hruza
;
Joon O. Jung
;
John K. F. Maclean
;
My Mansueto
;
George N. Naumov
;
Ulrike Philippar
;
Shruti Raut
;
Peter Spacciapoli
;
Dongyu Sun
;
Phieng Siliphaivanh
刊名:Journal of Medicinal Chemistry
出版年:20
1
6
4.
Phosphoproteome Profiling Reveals Molecular Mechanisms of Growth-Factor-Mediated
Kinase
Inhibitor Resistance in EGFR-Overexpressing Cancer Cells
作者:
Heiner Koch
;
Mathias Wilhelm
;
Benjamin Ruprecht
;
Scarlet Beck
;
Martin Frejno
;
Susan Klaeger
;
Bernhard Kuster
刊名:Journal of Proteome Research
出版年:20
1
6
5.
Human ATP-Binding Cassette Transporter ABCG2 Confers Resistance to CUDC-907, a Dual Inhibitor of Histone Deacetylase and Phosphatidylinositol 3-
Kinase
作者:
Chung-Pu Wu
;
Ya-Ju Hsieh
;
Sung-Han Hsiao
;
Ching-Ya Su
;
Yan-Qing Li
;
Yang-Hui Huang
;
Chiun-Wei Huang
;
Chia-Hung Hsieh
;
Jau-Song Yu
;
Yu-Shan Wu
刊名:Molecular Pharmaceutics
出版年:20
1
6
6.
Phosphorylation or Mutation of the ERK2 Activation Loop Alters Oligonucleotide Binding
作者:
Andrea C. McReynolds
;
Aroon S. Karra
;
Yan Li
;
Elias Daniel Lopez
;
Adrian G. Turjanski
;
Elhadji Dioum
;
Kristina Lorenz
;
Elma Zaganjor
;
Steve Stippec
;
Kathleen McGlynn
;
Svetlana Earnest
;
Melanie H. Cobb
刊名:Biochemistry
出版年:20
1
6
7.
MAP4K4 Is a Threonine
Kinase
That Phosphorylates FARP
1
作者:
Adam G. Schwaid
;
Chunyan Su
;
Paula Loos
;
Jiang Wu
;
Chuong Nguyen
;
Kathryn L. Stone
;
Jean Kanyo
;
Kieran F. Geoghegan
;
Samit K. Bhattacharya
;
Robert L. Dow
;
Leonard Buckbinder
;
Philip A. Carpino
刊名:ACS Chemical Biology
出版年:20
1
5
8.
Discovery and Optimization of a Novel Series of Dyrk
1
B
Kinase
Inhibitors To Explore a
MEK
Resistance Hypothesis
作者:
Jason G. Kettle
;
Peter Ballard
;
Catherine Bardelle
;
Mark Cockerill
;
Nicola Colclough
;
Susan E. Critchlow
;
Judit Debreczeni
;
Gary Fairley
;
Shaun Fillery
;
Mark A. Graham
;
Louise Goodwin
;
Sylvie Guichard
;
Kevin Hudson
;
Richard A. Ward
;
David Whittaker
刊名:Journal of Medicinal Chemistry
出版年:20
1
5
9.
SUN
11
602, a Novel Aniline Compound, Mimics the Neuroprotective Mechanisms of Basic Fibroblast Growth Factor
作者:
Norihito Murayama
;
Taisuke Kadoshima
;
Naohiro Takemoto
;
Shiho Kodama
;
Tetsuya Toba
;
Ryoko Ogino
;
Takafumi Noshita
;
Tetsushi Oka
;
Shinya Ueno
;
Mariko Kuroda
;
Yoshiari Shimmyo
;
Yasuhiro Morita
;
Teruyoshi Inoue
刊名:ACS Chemical Neuroscience
出版年:20
1
3
10.
Novel 3-Substituted 7-Phenylpyrrolo[3,2-f]quinolin-9(6H)-ones as Single Entities with Multitarget Antiproliferative Activity
作者:
Davide Carta
;
Roberta Bortolozzi
;
Ernest Hamel
;
Giuseppe Basso
;
Stefano Moro
;
Giampietro Viola
;
Maria Grazia Ferlin
刊名:Journal of Medicinal Chemistry
出版年:20
1
5
1
2
3
4
5
6
7
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